Document Detail


The toxicokinetics of (1R, cis)- and (1R, trans)- tetramethrin in the isolated perfused rat liver.
MedLine Citation:
PMID:  2750207     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
1. The toxicokinetics of cis- and trans-tetramethrin isomers were investigated using the isolated perfused rat liver preparation. 2. The concentration of cis- and trans-tetramethrin decreased rapidly in the plasma perfusate and was initially replaced by N-(hydroxymethyl)3,4,5,6-tetrahydrophthalimide (MTI) and then by 3,4,5,6-tetrahydrophthalimide (TPI). Plasma perfusate concentrations of the intact cis-isomer were higher than those of the trans-isomer. Concentrations of MTI and TPI were higher in livers treated with the trans-isomer. 3. Tetramethrin and its metabolites were rapidly excreted in the bile. Bile from livers perfused with trans-isomer contained higher concentrations of parent isomer and metabolites MTI and TPI, than did bile from livers treated with the cis-isomer.
Authors:
I S Silver; W C Dauterman
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Publication Detail:
Type:  In Vitro; Journal Article; Research Support, U.S. Gov't, P.H.S.    
Journal Detail:
Title:  Xenobiotica; the fate of foreign compounds in biological systems     Volume:  19     ISSN:  0049-8254     ISO Abbreviation:  Xenobiotica     Publication Date:  1989 May 
Date Detail:
Created Date:  1989-08-25     Completed Date:  1989-08-25     Revised Date:  2007-11-15    
Medline Journal Info:
Nlm Unique ID:  1306665     Medline TA:  Xenobiotica     Country:  ENGLAND    
Other Details:
Languages:  eng     Pagination:  509-19     Citation Subset:  IM    
Affiliation:
Toxicology Program, North Carolina State University, Raleigh 27695.
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MeSH Terms
Descriptor/Qualifier:
Animals
Bile / metabolism
Captan
Kinetics
Liver / drug effects,  metabolism*
Male
Perfusion
Phthalimides / metabolism
Pyrethrins / metabolism*,  toxicity
Rats
Rats, Inbred Strains
Stereoisomerism
Grant Support
ID/Acronym/Agency:
ES-00044/ES/NIEHS NIH HHS; ES-07046/ES/NIEHS NIH HHS
Chemical
Reg. No./Substance:
0/Phthalimides; 0/Pyrethrins; 133-06-2/Captan; 27813-21-4/tetrahydrophthalimide; 7696-12-0/tetramethrin

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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