Document Detail


A safer methylation procedure with boron trifluoride-methanol reagent for gas chromatographic analysis of ritalinic acid in urine.
MedLine Citation:
PMID:  1391098     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Ritalinic acid (RITA), the major metabolite of methylphenidate (Ritaline) is extracted with a solid-phase C8 column. Following elution, methylation of the carboxylic group is performed with boron trifluoride-methanol as a reagent. The methyl ester of RITA which structurally corresponds to the parent compound methylphenidate is reextracted at pH 9-11. Each step of the analytical method has been systematically studied, particularly the parameters governing the esterification reaction with BF3-methanol. The recovery from the overall method is 96%. The limit of detection is 0.05 micrograms ml-1 with GC-NPD for a 10-ml urine sample. The method has been successfully applied to the detection and quantitation of RITA in urine specimens. The specificity of the methylated RITA peak has been verified by GC-MS in scan mode. Use of diazomethane or sulphuric acid is thus replaced by the use of a less hazardous reagent.
Authors:
T Vu-Duc; A Vernay
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Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Journal of pharmaceutical and biomedical analysis     Volume:  10     ISSN:  0731-7085     ISO Abbreviation:  J Pharm Biomed Anal     Publication Date:    1992 Feb-Mar
Date Detail:
Created Date:  1992-10-29     Completed Date:  1992-10-29     Revised Date:  2004-11-17    
Medline Journal Info:
Nlm Unique ID:  8309336     Medline TA:  J Pharm Biomed Anal     Country:  ENGLAND    
Other Details:
Languages:  eng     Pagination:  187-91     Citation Subset:  IM    
Affiliation:
Unit of Drug Analysis, Institute of Occupational Health Sciences, Lausanne, Switzerland.
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MeSH Terms
Descriptor/Qualifier:
Boranes / chemistry*
Chromatography, Gas
Humans
Indicators and Reagents / chemistry
Methanol / chemistry*
Methylation
Methylphenidate / analogs & derivatives*,  metabolism,  urine
Temperature
Chemical
Reg. No./Substance:
0/Boranes; 0/Indicators and Reagents; 113-45-1/Methylphenidate; 19395-41-6/ritalinic acid; 67-56-1/Methanol; 7637-07-2/boron trifluoride

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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