Document Detail


A prolyl oligopeptidase inhibitor, Z-Pro-Prolinal, inhibits glyceraldehyde-3-phosphate dehydrogenase translocation and production of reactive oxygen species in CV1-P cells exposed to 6-hydroxydopamine.
MedLine Citation:
PMID:  16942854     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
We studied the ability of prolyl oligopeptidase (POP) inhibitors, Z-Pro-Prolinal and JTP-4819, to prevent translocation of glyceraldehyde-3-phosphate dehydrogenase (GAPDH) and formation of reactive oxygen species (ROS), in 6-hydroxydopamine (6-OHDA) and cytosine arabinoside (Ara-C) treated monkey fibroblast (CV1-P) and human neuroblastoma (SH-SY5Y) cells. The cells were pretreated with POP inhibitors (30 min) before addition of toxicants. GAPDH was analyzed by Western hybridization, ROS by fluorescent 2'7'-dichlorodihydro-fluorescein diacetate, and viability by the MTT method. Both toxicants induced GAPDH translocation to the particulate fraction (mitochondria and nuclei). Z-Pro-Prolinal was able to inhibit the translocation in 6-OHDA-exposed CV1-P cells. In SH-SY5Y cells and in JTP-4819 pretreated cells, no prevention of translocation was seen. However, the intensity of GAPDH in cytosolic fraction increased. Both inhibitors blocked 6-OHDA-induced ROS-production to the control level in CV1-P but, not in SH-SY5Y cells, without affecting their viability. In conclusion, POP inhibitors are able to prevent certain cell stress related factors such as ROS production or GAPDH translocation.
Authors:
Katja A Puttonen; Sárka Lehtonen; Atso Raasmaja; Pekka T Männistö
Related Documents :
10498294 - Reactive oxygen species production by monoamine oxidases in intact cells.
17412404 - Cross-reactivity patterns of t cells specific for iodinated contrast media.
19298354 - Photodynamic inactivation of candida albicans by bam-sipc.
3165394 - Peripheral pmn cells in juvenile periodontitis. increased release of elastase and of ox...
6365644 - Insulin release : the fuel concept.
3118984 - A cell-free analysis of the endocytic pathway.
Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't     Date:  2006-07-14
Journal Detail:
Title:  Toxicology in vitro : an international journal published in association with BIBRA     Volume:  20     ISSN:  0887-2333     ISO Abbreviation:  Toxicol In Vitro     Publication Date:  2006 Dec 
Date Detail:
Created Date:  2006-10-18     Completed Date:  2006-12-26     Revised Date:  2009-04-10    
Medline Journal Info:
Nlm Unique ID:  8712158     Medline TA:  Toxicol In Vitro     Country:  England    
Other Details:
Languages:  eng     Pagination:  1446-54     Citation Subset:  IM    
Affiliation:
Department of Pharmacology and Toxicology, University of Kuopio, P.O. Box 1627, FIN-70211 Kuopio, Finland. katja.puttonen@uku.fi
Export Citation:
APA/MLA Format     Download EndNote     Download BibTex
MeSH Terms
Descriptor/Qualifier:
Actins / biosynthesis,  genetics
Blotting, Western
Cell Line
Cell Survival / drug effects
Cytarabine / antagonists & inhibitors,  toxicity
Dipeptides / pharmacology*
Glyceraldehyde-3-Phosphate Dehydrogenases / metabolism*
Humans
Oxidopamine / antagonists & inhibitors*,  toxicity*
Protease Inhibitors / pharmacology*
Protein Transport / drug effects
Proto-Oncogene Proteins c-bcl-2 / metabolism
Pyrrolidines / pharmacology
Reactive Oxygen Species / metabolism*
Serine Endopeptidases / metabolism*
Tetrazolium Salts
Thiazoles
Tumor Suppressor Protein p53 / metabolism
Chemical
Reg. No./Substance:
0/Actins; 0/Dipeptides; 0/JTP 4819; 0/Protease Inhibitors; 0/Proto-Oncogene Proteins c-bcl-2; 0/Pyrrolidines; 0/Reactive Oxygen Species; 0/Tetrazolium Salts; 0/Thiazoles; 0/Tumor Suppressor Protein p53; 1199-18-4/Oxidopamine; 147-94-4/Cytarabine; 298-93-1/thiazolyl blue; 86925-97-5/N-benzyloxycarbonylprolylprolinal; EC 1.2.1.-/Glyceraldehyde-3-Phosphate Dehydrogenases; EC 3.4.21.-/Serine Endopeptidases; EC 3.4.21.26/prolyl oligopeptidase

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


Previous Document:  In vitro biological efficiency of tenocyclidine-TCP and its adamantane derivative TAMORF.
Next Document:  The human basonuclin 2 gene has the potential to generate nearly 90,000 mRNA isoforms encoding over ...