Document Detail


p53 and TIGAR regulate cardiac myocyte energy homeostasis under hypoxic stress.
MedLine Citation:
PMID:  20935145     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Bioenergetic homeostasis is altered in heart failure and may play an important role in pathogenesis. p53 has been implicated in heart failure, and although its role in regulating tumorigenesis is well characterized, its activities on cellular metabolism are just beginning to be understood. We investigated the role of p53 and its transcriptional target gene TP53-induced glycolysis and apoptosis regulator (TIGAR) in myocardial energy metabolism under conditions simulating ischemia that can lead to heart failure. Expression of p53 and TIGAR was markedly upregulated after myocardial infarction, and apoptotic myocytes were decreased by 42% in p53-deficient mouse hearts compared with those in wild-type mice. To examine the effect of p53 on energy metabolism, cardiac myocytes were exposed to hypoxia. Hypoxia induced p53 and TIGAR expression in a p53-dependent manner. Knockdown of p53 or TIGAR increased glycolysis with elevated fructose-2,6-bisphosphate levels and reduced myocyte apoptosis. Hypoxic stress decreased phosphocreatine content and the mitochondrial membrane potential of myocytes without changes in ATP content, the effects of which were prevented by the knockdown of TIGAR. Inhibition of glycolysis by 2-deoxyglucose blocked these bioenergetic effects and TIGAR siRNA-mediated prevention of apoptosis, and, in contrast, overexpression of TIGAR reduced glucose utilization and increased apoptosis. Our data demonstrate that p53 and TIGAR inhibit glycolysis in hypoxic myocytes and that inhibition of glycolysis is closely involved in apoptosis, suggesting that p53 and TIGAR are significant mediators of cellular energy homeostasis and cell death under ischemic stress.
Authors:
Masaki Kimata; Satoaki Matoba; Eri Iwai-Kanai; Hideo Nakamura; Atsushi Hoshino; Mikihiko Nakaoka; Maki Katamura; Yoshifumi Okawa; Yuichiro Mita; Mitsuhiko Okigaki; Koji Ikeda; Tetsuya Tatsumi; Hiroaki Matsubara
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't     Date:  2010-10-08
Journal Detail:
Title:  American journal of physiology. Heart and circulatory physiology     Volume:  299     ISSN:  1522-1539     ISO Abbreviation:  Am. J. Physiol. Heart Circ. Physiol.     Publication Date:  2010 Dec 
Date Detail:
Created Date:  2010-12-03     Completed Date:  2011-01-13     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  100901228     Medline TA:  Am J Physiol Heart Circ Physiol     Country:  United States    
Other Details:
Languages:  eng     Pagination:  H1908-16     Citation Subset:  IM    
Affiliation:
Department of Cardiovascular Medicine, Kyoto Prefectural University School of Medicine, Kyoto, Japan.
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MeSH Terms
Descriptor/Qualifier:
Adenosine Triphosphate / metabolism
Animals
Apoptosis
Apoptosis Regulatory Proteins / genetics,  metabolism*
Cell Hypoxia
Cells, Cultured
Deoxyglucose / metabolism
Disease Models, Animal
Energy Metabolism*
Glycolysis
Homeostasis
Membrane Potential, Mitochondrial
Mice
Mice, Knockout
Myocardial Infarction / genetics,  metabolism*,  pathology
Myocytes, Cardiac / metabolism*,  pathology
Phosphocreatine / metabolism
Phosphofructokinase-2 / metabolism
Proteins / genetics,  metabolism*
RNA Interference
Rats
Stress, Physiological*
Time Factors
Transfection
Tumor Suppressor Protein p53 / deficiency,  genetics,  metabolism*
Chemical
Reg. No./Substance:
0/Apoptosis Regulatory Proteins; 0/Proteins; 0/TIGAR protein, mouse; 0/Tumor Suppressor Protein p53; 154-17-6/Deoxyglucose; 56-65-5/Adenosine Triphosphate; 67-07-2/Phosphocreatine; EC 2.7.1.105/Phosphofructokinase-2

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