Document Detail


The emerging role of serine proteases in apoptosis.
MedLine Citation:
PMID:  17511651     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Unregulated apoptosis can be due to a disruption in the balance and control of both intra- and inter-cellular proteolytic activities leading to various disease states. Many proteases involved in apoptotic processes are yet to be identified; however, several are already well characterized. Caspases traditionally held the predominant role as prime mediators of execution. However, latterly, evidence has accumulated that non-caspases, including calpains, cathepsins, granzymes and the proteasome have roles in mediating and promoting cell death. Increasingly, research is implicating serine proteases within apoptotic processing, particularly in the generation of nuclear events such as condensation, fragmentation and DNA degradation observed in late-stage apoptosis. Serine proteases therefore are emerging as providing additional or alternative therapeutic targets.
Authors:
K L Moffitt; S L Martin; B Walker
Publication Detail:
Type:  Journal Article; Review    
Journal Detail:
Title:  Biochemical Society transactions     Volume:  35     ISSN:  0300-5127     ISO Abbreviation:  Biochem. Soc. Trans.     Publication Date:  2007 Jun 
Date Detail:
Created Date:  2007-05-21     Completed Date:  2007-08-06     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  7506897     Medline TA:  Biochem Soc Trans     Country:  England    
Other Details:
Languages:  eng     Pagination:  559-60     Citation Subset:  IM    
Affiliation:
School of Pharmacy, Queen's University, Belfast BT9 7BL, Northern Ireland, UK. kellylmoffitt@hotmail.com
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MeSH Terms
Descriptor/Qualifier:
Animals
Apoptosis / physiology*
Granzymes / metabolism
Humans
Mitochondrial Proteins / metabolism
Serine Endopeptidases / metabolism*
Serpins / metabolism
Thrombin / metabolism
Chemical
Reg. No./Substance:
0/Mitochondrial Proteins; 0/Serpins; EC 3.4.21.-/AP24 apoptotic protease; EC 3.4.21.-/Granzymes; EC 3.4.21.-/Omi serine protease; EC 3.4.21.-/Serine Endopeptidases; EC 3.4.21.5/Thrombin

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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