Document Detail


An efficient pH sensitive oral insulin delivery system enhanced by deoxycholic acid.
MedLine Citation:
PMID:  22195840     Owner:  NLM     Status:  In-Data-Review    
Abstract/OtherAbstract:
A permeation enhancer, positively charged deoxycholyl-hyperbranched oligoethylenimine (DCO), was prepared and used to form complexes with negatively charged insulin based on electrostatic interaction. DCO/insulin complexes can be loaded into poly (l-glutamic acid) (PGA) microspheres by the oil-in-oil (O/O) emulsion and solvent evaporation technique. Because of the specific pH sensitive properties of PGA, these insulin encapsulated microspheres are stable in the stomach and disaggregate in the small intestine, and the bioavailability of oral insulin administration will be improved due to DCO's permeation enhancement function.
Authors:
Li Zhao; Jianxun Ding; Pan He; Chunsheng Xiao; Zhaohui Tang; Xiuli Zhuang; Xuesi Chen
Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Journal of controlled release : official journal of the Controlled Release Society     Volume:  152 Suppl 1     ISSN:  1873-4995     ISO Abbreviation:  J Control Release     Publication Date:  2011 Nov 
Date Detail:
Created Date:  2011-12-26     Completed Date:  -     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  8607908     Medline TA:  J Control Release     Country:  Netherlands    
Other Details:
Languages:  eng     Pagination:  e184-6     Citation Subset:  IM    
Copyright Information:
Copyright © 2011. Published by Elsevier B.V.
Affiliation:
Key Laboratory of Polymer Ecomaterials, Changchun Institute of Applied Chemistry, Chinese Academy of Sciences, Changchun 130022, China; Graduate University of the Chinese Academy of Sciences, Beijing 100039, China.
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