Document Detail


The effects in myometrial preparations of D2343, a beta 2-adrenoceptor agonist possessing alpha 1-receptor blocking qualities.
MedLine Citation:
PMID:  6152105     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
D2343 is a compound with about the same beta 2-adrenoceptor-agonist effect as terbutaline and exhibiting in addition an alpha 1-receptor inhibitory activity. D2343 has been compared to the beta 2-agonist terbutaline on oestrogenized uterine preparations from rat and rabbit (in vitro and in vivo) and in myometrial strips from homo. Generally, D2343 has shown an ability to relax the uterine muscles to the same degree as terbutaline or even more, especially when the two drugs were compared in vitro in preparations from rabbit and rat.
Authors:
O A Olsson; B Ahlquist; B Gustafsson; G Persson
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Publication Detail:
Type:  Comparative Study; In Vitro; Journal Article    
Journal Detail:
Title:  Acta pharmacologica et toxicologica     Volume:  55     ISSN:  0001-6683     ISO Abbreviation:  Acta Pharmacol Toxicol (Copenh)     Publication Date:  1984 Nov 
Date Detail:
Created Date:  1985-04-15     Completed Date:  1985-04-15     Revised Date:  2006-11-15    
Medline Journal Info:
Nlm Unique ID:  0370572     Medline TA:  Acta Pharmacol Toxicol (Copenh)     Country:  DENMARK    
Other Details:
Languages:  eng     Pagination:  391-7     Citation Subset:  IM    
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MeSH Terms
Descriptor/Qualifier:
Adrenergic alpha-Antagonists / pharmacology*
Adrenergic beta-Agonists / pharmacology*
Animals
Carbachol / antagonists & inhibitors
Estradiol / pharmacology
Female
Humans
Octopamine / analogs & derivatives*,  pharmacology
Oxytocin / antagonists & inhibitors
Rabbits
Rats
Rats, Inbred Strains
Terbutaline / pharmacology
Uterine Contraction / drug effects*
Chemical
Reg. No./Substance:
0/Adrenergic alpha-Antagonists; 0/Adrenergic beta-Agonists; 104-14-3/Octopamine; 23031-25-6/Terbutaline; 50-28-2/Estradiol; 50-56-6/Oxytocin; 51-83-2/Carbachol; 72734-63-5/D 2343

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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