Document Detail


The effect of proadifen, a drug metabolism inhibitor, on action of imipramine and desipramine in mice.
MedLine Citation:
PMID:  7187047     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Proadifen (SKF 524 A) inhibited the following effects of imipramine (IMI), without affecting those of desipramine (DMI) in mice: antagonism towards reserpine-induced hypothermia, ptosis and sedation, antagonism to apomorphine hypothermia and insignificant shortening of the immobility time in the behavioral despair test. Cerebral levels of DMI were very low after administration of IMI; pretreatment with proadifen did not affect the already low levels of DMI but significantly elevated these of IMI. This may indicate that some other than DMI metabolites (e.g., 2-hydroxy-derivatives) may be of importance for the action of IMI in mice in the tests employed in this study.
Authors:
J Maj; M Melzacka; Z Rogóz; G Skuza; H Sowińska
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Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Polish journal of pharmacology and pharmacy     Volume:  34     ISSN:  0301-0244     ISO Abbreviation:  Pol J Pharmacol Pharm     Publication Date:    1982 Nov-Dec
Date Detail:
Created Date:  1983-12-20     Completed Date:  1983-12-20     Revised Date:  2003-11-14    
Medline Journal Info:
Nlm Unique ID:  0366561     Medline TA:  Pol J Pharmacol Pharm     Country:  POLAND    
Other Details:
Languages:  eng     Pagination:  323-31     Citation Subset:  IM    
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MeSH Terms
Descriptor/Qualifier:
Animals
Apomorphine / pharmacology
Behavior, Animal / drug effects
Blepharoptosis / chemically induced
Body Temperature / drug effects
Brain Chemistry / drug effects
Desipramine / antagonists & inhibitors*
Hypnotics and Sedatives
Imipramine / antagonists & inhibitors*
Male
Mice
Proadifen / pharmacology*
Reserpine / pharmacology
Chemical
Reg. No./Substance:
0/Hypnotics and Sedatives; 302-33-0/Proadifen; 50-47-5/Desipramine; 50-49-7/Imipramine; 50-55-5/Reserpine; 58-00-4/Apomorphine

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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