Document Detail


The determination of trimazosin and its metabolite CP23445 in whole blood by high performance liquid chromatography using fluorescence detection.
MedLine Citation:
PMID:  6536811     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
A sensitive and specific assay for trimazosin and its metabolite CP23445 is described. The method employs reverse-phase high performance liquid chromatography (HPLC) with fluorescence detection. The limit of detection of the assay is 1 ng/ml whole blood for trimazosin and 0.5 ng/ml for CP23445. The coefficient of variation for trimazosin and CP23445 over a typical calibration size is 5.4% and 4.9%, respectively. Various drugs that may be coadministered with trimazosin are shown not to interfere in the assay. The method has been extensively employed to study the pharmacokinetics of trimazosin and CP23445, both in man and in animals.
Authors:
M A Hughes; P A Meredith; H L Elliott
Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Journal of pharmacological methods     Volume:  12     ISSN:  0160-5402     ISO Abbreviation:  J Pharmacol Methods     Publication Date:  1984 Aug 
Date Detail:
Created Date:  1985-09-16     Completed Date:  1985-09-16     Revised Date:  2004-11-17    
Medline Journal Info:
Nlm Unique ID:  7806596     Medline TA:  J Pharmacol Methods     Country:  UNITED STATES    
Other Details:
Languages:  eng     Pagination:  29-34     Citation Subset:  IM    
Export Citation:
APA/MLA Format     Download EndNote     Download BibTex
MeSH Terms
Descriptor/Qualifier:
Chromatography, High Pressure Liquid
Humans
Metabolic Clearance Rate
Piperazines / blood*,  metabolism
Spectrometry, Fluorescence
Chemical
Reg. No./Substance:
0/Piperazines; 35795-16-5/trimazosin; 88321-10-2/1-hydroxytrimazosin

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


Previous Document:  Alloimmune hemagglutinating antibodies in cynomolgus monkeys.
Next Document:  Determination of inflamed paw surface temperature in rats.