Document Detail


The decrease in uroporphyrinogen decarboxylase activity induced by ethanol predisposes rats to the development of porphyria and accelerates xenobiotic-triggered porphyria, regardless of hepatic damage.
MedLine Citation:
PMID:  12426626     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
We evaluated the porphyrinogenic ability of ethanol (20% in drinking water) per se, its effect on the development of sporadic porphyria cutanea tarda induced by hexachlorobenzene in female Wistar rats (170-190 g, N = 8/group), and the relationship with hepatic damage. Twenty-five percent of the animals receiving ethanol increased up to 14-, 25-, and 4.5-fold the urinary excretion of delta-aminolevulinate, porphobilinogen, and porphyrins, respectively. Ethanol exacerbated the precursor excretions elicited by hexachlorobenzene. Hepatic porphyrin levels increased by hexachlorobenzene treatment, while this parameter only increased (up to 90-fold) in some of the animals that received ethanol alone. Ethanol reduced the activities of uroporphyrinogen decarboxylase, delta-aminolevulinate dehydrase and ferrochelatase. In the ethanol group, many of the animals showed a 30% decrease in uroporphyrinogen activity; in the ethanol + hexachlorobenzene group, this decrease occurred before the one caused by hexachlorobenzene alone. Ethanol exacerbated the effects of hexachlorobenzene, among others, on the rate-limiting enzyme delta-aminolevulinate synthetase. The plasma activities of enzymes that are markers of hepatic damage were similar in all drug-treated groups. These results indicate that 1) ethanol exacerbates the biochemical manifestation of sporadic hexachlorobenzene-induced porphyria cutanea tarda; 2) ethanol per se affects several enzymatic and excretion parameters of the heme metabolic pathway; 3) since not all the animals were affected to the same extent, ethanol seems to be a porphyrinogenic agent only when there is a predisposition, and 4) hepatic damage showed no correlation with the development of porphyria cutanea tarda.
Authors:
M C Ríos de Molina; M B Mazzetti; M Galigniana; C Aldonatti; J M Tomio; L C San Martín de Viale
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  Brazilian journal of medical and biological research = Revista brasileira de pesquisas médicas e biológicas / Sociedade Brasileira de Biofísica ... [et al.]     Volume:  35     ISSN:  0100-879X     ISO Abbreviation:  Braz. J. Med. Biol. Res.     Publication Date:  2002 Nov 
Date Detail:
Created Date:  2002-11-11     Completed Date:  2003-04-02     Revised Date:  2006-11-15    
Medline Journal Info:
Nlm Unique ID:  8112917     Medline TA:  Braz J Med Biol Res     Country:  Brazil    
Other Details:
Languages:  eng     Pagination:  1273-83     Citation Subset:  IM    
Affiliation:
Laboratorio de Porfirias Experimentales y Metabolismo del Hemo, Departamento de Química Biológica, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires, Buenos Aires, Argentina.
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MeSH Terms
Descriptor/Qualifier:
Animals
Cytochrome P-450 Enzyme System / analysis
Disease Models, Animal
Ethanol / pharmacology*
Female
Ferrochelatase / drug effects*,  metabolism
Hexachlorobenzene
Liver / drug effects*,  enzymology,  pathology
Porphobilinogen / urine
Porphobilinogen Synthase / urine
Porphyria Cutanea Tarda / chemically induced*,  enzymology,  urine
Porphyrins / urine
Rats
Rats, Wistar
Solvents / pharmacology*
Uroporphyrinogen Decarboxylase / drug effects*,  metabolism
Chemical
Reg. No./Substance:
0/Porphyrins; 0/Solvents; 118-74-1/Hexachlorobenzene; 487-90-1/Porphobilinogen; 64-17-5/Ethanol; 9035-51-2/Cytochrome P-450 Enzyme System; EC 4.1.1.37/Uroporphyrinogen Decarboxylase; EC 4.2.1.24/Porphobilinogen Synthase; EC 4.99.1.1/Ferrochelatase

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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