Document Detail


The chlorophyll metabolite phytanic acid is a natural rexinoid--potential for treatment and prevention of diabetes.
MedLine Citation:
PMID:  11425290     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Synthetic ligands of the retinoid X receptor (RXR) have shown antidiabetic activity in mice, apparently owing to the fact that they stimulate the transcriptional activity of PPAR-gamma/RXR heterodimers, much like thiazolidinedione drugs. The chlorophyll metabolite phytanic acid has been shown to be a natural ligand for RXR, active in concentrations near its physiological levels. It is thus reasonable to suspect that phytanic acid may have utility for treatment and prevention of human type 2 diabetes. Phytanic acid may mimic or complement various effects of conjugated linoleic acids, which have been shown to activate PPAR-gamma/RXR and prevent rodent diabetes. Administration of hydrolyzed chlorophyll may represent the most cost-effective strategy for raising human tissue levels of phytanic acid.
Authors:
M F McCarty
Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Medical hypotheses     Volume:  56     ISSN:  0306-9877     ISO Abbreviation:  Med. Hypotheses     Publication Date:  2001 Feb 
Date Detail:
Created Date:  2001-06-29     Completed Date:  2001-08-02     Revised Date:  2004-11-17    
Medline Journal Info:
Nlm Unique ID:  7505668     Medline TA:  Med Hypotheses     Country:  Scotland    
Other Details:
Languages:  eng     Pagination:  217-9     Citation Subset:  IM    
Affiliation:
Pantox Laboratories, 4622 Santa Fe Street, San Diego, CA 92109, USA.
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MeSH Terms
Descriptor/Qualifier:
Animals
Chlorophyll / metabolism*
Diabetes Mellitus, Type 2 / prevention & control*
Humans
Linoleic Acid / pharmacology
Mice
Phytanic Acid / pharmacology,  therapeutic use*
Receptors, Cytoplasmic and Nuclear / drug effects
Transcription Factors / drug effects
Chemical
Reg. No./Substance:
0/Receptors, Cytoplasmic and Nuclear; 0/Transcription Factors; 1406-65-1/Chlorophyll; 14721-66-5/Phytanic Acid; 2197-37-7/Linoleic Acid

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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