Document Detail


Varenicline: progress in smoking cessation treatment.
MedLine Citation:
PMID:  17685891     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Varenicline is the first pharmacological aid for smoking cessation treatment to be approved in almost a decade. Varenicline is an alpha4beta2 nicotinic acetylcholine receptor partial agonist. It may assist those who wish to quit smoking by producing partial activation at nicotinic receptors to ease craving and withdrawal symptoms; and by simultaneously blocking the effects of nicotine from cigarettes smoked, thereby reducing the satisfaction of continued smoking. The effectiveness of varenicline as an aid for smoking cessation has been demonstrated in several clinical trials versus placebo and sustained release bupropion. In addition, varenicline is well tolerated and has an acceptable safety profile. As an aid for smoking cessation, varenicline offers progress in the treatment of tobacco dependence.
Authors:
Elbert D Glover; Jessica M Rath
Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't; Review    
Journal Detail:
Title:  Expert opinion on pharmacotherapy     Volume:  8     ISSN:  1744-7666     ISO Abbreviation:  Expert Opin Pharmacother     Publication Date:  2007 Aug 
Date Detail:
Created Date:  2007-08-09     Completed Date:  2007-09-17     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  100897346     Medline TA:  Expert Opin Pharmacother     Country:  England    
Other Details:
Languages:  eng     Pagination:  1757-67     Citation Subset:  IM    
Affiliation:
University of Maryland College Park School of Public Health, Department of Public & Community Health, College Park, MD 20742, USA. eglover1@umd.edu
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MeSH Terms
Descriptor/Qualifier:
Animals
Benzazepines / metabolism,  therapeutic use*
Humans
Quinoxalines / metabolism,  therapeutic use*
Receptors, Nicotinic / metabolism
Smoking / drug therapy*,  metabolism,  trends*
Smoking Cessation / methods*
Chemical
Reg. No./Substance:
0/Benzazepines; 0/Quinoxalines; 0/Receptors, Nicotinic; 0/varenicline

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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