Document Detail


Urocortin protects against ischemic injury via a MAPK-dependent pathway.
MedLine Citation:
PMID:  11597826     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Urocortin (UCN), is a peptide related to hypothalamic corticotrophin releasing hormone (CRF) and binds with high affinity to the CRF-R2 beta receptor which is expressed in the heart. UCN prevents cell death when administered to primary cardiac myocyte cultures both prior to simulated hypoxia/ischemia and at the point of reoxygenation after simulated hypoxia/ischemia as assayed by trypan blue exclusion. 3'-OH end labeling of DNA (TUNEL), annexin-V and fluorescence activated cell sorting. The protective effect of UCN is dependent on the p42/p44 mitogen-activated protein kinase (MAPK)-pathway. UCN also reduces damage in isolated rat hearts ex vivo, subjected to regional ischemia/reperfusion with the protective effect being observed when UCN is given either prior to ischemia or at the time of reperfusion after ischemia. Hence, UCN is a cardioprotective agent, which acts when given prior to ischemia or after ischemia at reperfusion.
Authors:
D S Latchman
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't; Review    
Journal Detail:
Title:  Trends in cardiovascular medicine     Volume:  11     ISSN:  1050-1738     ISO Abbreviation:  Trends Cardiovasc. Med.     Publication Date:  2001 Jul 
Date Detail:
Created Date:  2001-10-12     Completed Date:  2001-12-04     Revised Date:  2009-11-19    
Medline Journal Info:
Nlm Unique ID:  9108337     Medline TA:  Trends Cardiovasc Med     Country:  United States    
Other Details:
Languages:  eng     Pagination:  167-9     Citation Subset:  IM    
Affiliation:
Institute of Child Health, University College London, London, United Kingdom.
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MeSH Terms
Descriptor/Qualifier:
Animals
Corticotropin-Releasing Hormone / metabolism*,  therapeutic use*
Mitogen-Activated Protein Kinases / metabolism*
Myocardial Ischemia / drug therapy,  metabolism,  prevention & control*
Protective Agents / metabolism*,  therapeutic use*
Rats
Receptors, Corticotropin-Releasing Hormone / metabolism
Urocortins
Chemical
Reg. No./Substance:
0/CRF receptor type 2; 0/Protective Agents; 0/Receptors, Corticotropin-Releasing Hormone; 0/Urocortins; 9015-71-8/Corticotropin-Releasing Hormone; EC 2.7.11.24/Mitogen-Activated Protein Kinases

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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