Document Detail


Telmisartan improves endothelial function in patients with essential hypertension.
MedLine Citation:
PMID:  18049303     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
BACKGROUND:: Hypertension is a cardiovascular risk factor commonly associated with endothelial dysfunction and increased renal vascular resistance. Angiotensin receptor blockers (ARBs) may beneficially affect these parameters via antagonism of angiotensin type 1 (AT1) receptor-mediated vasoconstriction and vascular superoxide production. We therefore investigated whether the new ARB telmisartan improves endothelial function and renal vascular resistance in patients with essential hypertension. METHODS:: Thirty-seven patients with essential hypertension were randomized to receive telmisartan, the calcium channel blocker nisoldipine, or their combination for 6 weeks in a prospective, parallel group study. Brachial artery flow-mediated (endothelium-dependent) dilation (FMD) and renal vascular resistance index (RVRI) were evaluated using high-resolution ultrasound before, at 3 weeks (low dose), and at 6 weeks (high dose) after initiation of treatment. RESULTS:: At baseline, FMD and RVRI did not significantly differ between treatment groups. After 3 weeks of treatment neither treatment significantly changed FMD or RVRI. After 6 weeks of treatment, patients randomized to receive telmisartan alone or the combination, but not those treated with nisoldipine alone, displayed a significantly improved FMD, whereas RVRI values again were not significantly different as compared to those at baseline. CONCLUSION:: In our study cohort of patients with essential hypertension, treatment with telmisartan improved FMD but did not change RVRI. Future studies will demonstrate whether this telmisartan-induced effect may contribute to a blood pressure-independent reduction in cardiovascular morbidity.
Authors:
Ralf A Benndorf; Daniel Appel; Renke Maas; Edzard Schwedhelm; Ulrich O Wenzel; Rainer H Böger
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Publication Detail:
Type:  Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  Journal of cardiovascular pharmacology     Volume:  50     ISSN:  0160-2446     ISO Abbreviation:  J. Cardiovasc. Pharmacol.     Publication Date:  2007 Oct 
Date Detail:
Created Date:  2007-11-30     Completed Date:  2008-02-05     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  7902492     Medline TA:  J Cardiovasc Pharmacol     Country:  United States    
Other Details:
Languages:  eng     Pagination:  367-71     Citation Subset:  IM    
Affiliation:
Clinical Pharmacology Unit, Institute of Experimental and Clinical Pharmacology, University Medical Center, Hamburg-Eppendorf, Germany. benndorf@uke.uni-hamburg.de
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MeSH Terms
Descriptor/Qualifier:
Aged
Angiotensin II Type 1 Receptor Blockers / pharmacology,  therapeutic use
Antihypertensive Agents / pharmacology,  therapeutic use
Benzimidazoles / pharmacology,  therapeutic use*
Benzoates / pharmacology,  therapeutic use*
Blood Pressure / drug effects
Drug Therapy, Combination
Endothelium, Vascular / drug effects*,  physiopathology
Female
Humans
Hypertension / drug therapy*
Kidney / blood supply,  drug effects
Male
Middle Aged
Nisoldipine / pharmacology,  therapeutic use
Prospective Studies
Single-Blind Method
Treatment Outcome
Vascular Resistance / drug effects
Vasodilation / drug effects
Chemical
Reg. No./Substance:
0/Angiotensin II Type 1 Receptor Blockers; 0/Antihypertensive Agents; 0/Benzimidazoles; 0/Benzoates; 144701-48-4/telmisartan; 63675-72-9/Nisoldipine

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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