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Synthesis, circular dichroism, and absolute stereochemistry of a Fecht acid analog and related compounds
MedLine Citation:
PMID:  10857059     Owner:  NLM     Status:  Publisher    
Abstract/OtherAbstract:
2,6-Dimethylspiro[3.3]heptane-2,6-dicarboxylic acid (2), an analog of the Fecht acid (1), was enantioresolved by the method of (1S,2R,4R)-(-)-2,10-camphorsultam yielding enantiopure acid (+)-2, the S absolute configuration of which was unambiguously determined by X-ray crystallography of camphorsultam amide derivative (R)-(-)-12b and chemical correlation. To determine the absolute configuration of chiral spiro[3.3]heptane compounds by the circular dichroism (CD) exciton chirality method, acid (+)-2 was converted to (+)-2,6-bis(phenylacetylenyl)-2,6-dimethylspiro[3.3]heptane (3) and (+)-2,6-bis(4-methoxyphenylacetylenyl)-2,6-dimethylspiro[3.3]heptane (4). The CD spectra of (+)-3 and (+)-4 exhibit intense exciton split Cotton effects of positive chirality, from which their S absolute configurations were confirmed.
Authors:
Murai; Soutome; Yoshida; Osawa; Harada
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Publication Detail:
Type:  JOURNAL ARTICLE    
Journal Detail:
Title:  Enantiomer     Volume:  5     ISSN:  1024-2430     ISO Abbreviation:  Enantiomer     Publication Date:  2000  
Date Detail:
Created Date:  2000-06-16     Completed Date:  -     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  9612491     Medline TA:  Enantiomer     Country:  ENGLAND    
Other Details:
Languages:  Eng     Pagination:  197-202     Citation Subset:  -    
Affiliation:
Institute for Chemical Reaction Science, Tohoku University, Sendai, Japan.
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