Document Detail


Synthesis of N-[tris[2-[[N-(benzyloxy)amino]carbonyl]ethyl]methyl]succinamic acid, trisuccin. Hydroxamic acid derivatives as a new class of bifunctional chelating agents.
MedLine Citation:
PMID:  8324008     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
In an effort to generate bifunctional chelating agents (BCAs) with improved labeling, conjugation, and biodistribution properties, the synthesis of trisuccin is reported. This new hydroxamate BCA, after synthesis and characterization, was used for conjugation and radiolabeling of monoclonal antibodies with 99mTc. This new class of synthetic BCAs may be useful in the radioimmunodiagnosis and radioimmunotherapy of cancer.
Authors:
A Safavy; D J Buchsbaum; M B Khazaeli
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Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Bioconjugate chemistry     Volume:  4     ISSN:  1043-1802     ISO Abbreviation:  Bioconjug. Chem.     Publication Date:    1993 May-Jun
Date Detail:
Created Date:  1993-08-09     Completed Date:  1993-08-09     Revised Date:  2000-12-18    
Medline Journal Info:
Nlm Unique ID:  9010319     Medline TA:  Bioconjug Chem     Country:  UNITED STATES    
Other Details:
Languages:  eng     Pagination:  194-8     Citation Subset:  IM    
Affiliation:
Department of Radiation Oncology, University of Alabama, Birmingham 35233.
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MeSH Terms
Descriptor/Qualifier:
Antibodies, Monoclonal
Chelating Agents / chemical synthesis*,  chemistry
Chromatography, Thin Layer
Cross-Linking Reagents / chemical synthesis*,  chemistry
Hydroxamic Acids / chemical synthesis*,  chemistry
Immunotoxins / chemistry
Isotope Labeling / methods
Magnetic Resonance Spectroscopy
Succinates / chemical synthesis*,  chemistry
Technetium / chemistry
Chemical
Reg. No./Substance:
0/Antibodies, Monoclonal; 0/Chelating Agents; 0/Cross-Linking Reagents; 0/Hydroxamic Acids; 0/Immunotoxins; 0/Succinates; 147219-26-9/trisuccin; 7440-26-8/Technetium

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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