Document Detail


Regulation of low-density lipoprotein receptor and 3-hydroxy-3-methylglutaryl coenzyme A reductase expression by Zingiber officinale in the liver of high-fat diet-fed rats.
MedLine Citation:
PMID:  20002065     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Zingiber officinale has been used to control lipid disorders and reported to possess remarkable cholesterol-lowering activity in experimental hyperlipidaemia. In the present study, the effect of a characterized and standardized extract of Zingiber officinale on the hepatic lipid levels as well as on the hepatic mRNA and protein expression of low-density lipoprotein (LDL) receptor and 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase was investigated in a high-fat diet-fed rat model. Rats were treated with an ethanol extract of Zingiber officinale (400 mg/kg) extract along with a high-fat diet for 6 weeks. The extract of Zingiber officinale significantly decreased hepatic triglyceride and tended to decrease hepatic cholesterol levels when administered over 6 weeks to the rats fed a high-fat diet. We found that in parallel, the extract up-regulated both LDL receptor mRNA and protein level and down-regulated HMG-CoA reductase protein expression in the liver of these rats. The metabolic control of body lipid homeostasis is in part due to enhanced cholesterol biosynthesis and reduced expression of LDL receptor sites following long-term consumption of high-fat diets. The present results show restoration of transcriptional and post-transcriptional changes in low-density lipoprotein and HMG CoA reductase by Zingiber officinale administration with a high-fat diet and provide a rational explanation for the effect of ginger in the treatment of hyperlipidaemia.
Authors:
Srinivas Nammi; Moon S Kim; Navnath S Gavande; George Q Li; Basil D Roufogalis
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't     Date:  2009-12-07
Journal Detail:
Title:  Basic & clinical pharmacology & toxicology     Volume:  106     ISSN:  1742-7843     ISO Abbreviation:  Basic Clin. Pharmacol. Toxicol.     Publication Date:  2010 May 
Date Detail:
Created Date:  2010-06-07     Completed Date:  2010-11-22     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  101208422     Medline TA:  Basic Clin Pharmacol Toxicol     Country:  Denmark    
Other Details:
Languages:  eng     Pagination:  389-95     Citation Subset:  IM    
Affiliation:
Herbal Medicines Research & Education Centre, Faculty of Pharmacy, University of Sydney, Sydney, NSW, Australia. snammi@pharm.usyd.edu.au
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MeSH Terms
Descriptor/Qualifier:
Animals
Cholesterol / metabolism
Diet
Dietary Fats / administration & dosage
Ethanol / chemistry
Fats / metabolism
Ginger / chemistry*
Hydroxymethylglutaryl CoA Reductases / biosynthesis,  genetics,  metabolism*
Lipoproteins, LDL / metabolism
Liver / drug effects*,  enzymology,  metabolism
Plant Extracts / chemistry,  pharmacology
RNA, Messenger / metabolism
Rats
Receptors, LDL / biosynthesis,  genetics,  metabolism*
Triglycerides / metabolism
Chemical
Reg. No./Substance:
0/Dietary Fats; 0/Fats; 0/Lipoproteins, LDL; 0/Plant Extracts; 0/RNA, Messenger; 0/Receptors, LDL; 0/Triglycerides; 57-88-5/Cholesterol; 64-17-5/Ethanol; EC 1.1.1.-/Hydroxymethylglutaryl CoA Reductases

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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