Document Detail


Regio- and stereo-selectivity in the induction of peroxisome proliferation by substituted hexanoic acids.
MedLine Citation:
PMID:  8518749     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Quantitative structure-activity relationship is an effective tool in order to predict drug potency. A similar approach is actually developed for peroxisome proliferation induced by substituted carboxylic acids issued from plasticizer metabolism in rats. The study is focused on acids found in rat urine after adipic diester dosings. Size, location of the substituted group and length of the chain have been studied. 3-D structure has also been taken in account for 2-ethyl hexanoic acids. The results obtained so far demonstrate that peroxisome proliferation potencies of the considered acids are modified according structure changes. At this time location of the group along the chain appears to be a predominant factor.
Authors:
A C Macherey; I Leguy; S Gregoire; G Tainturier; J C Lhuguenot
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Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Biology of the cell / under the auspices of the European Cell Biology Organization     Volume:  77     ISSN:  0248-4900     ISO Abbreviation:  Biol. Cell     Publication Date:  1993  
Date Detail:
Created Date:  1993-07-29     Completed Date:  1993-07-29     Revised Date:  2003-11-14    
Medline Journal Info:
Nlm Unique ID:  8108529     Medline TA:  Biol Cell     Country:  FRANCE    
Other Details:
Languages:  eng     Pagination:  9-11     Citation Subset:  IM    
Affiliation:
ENS BANA, Université de Bourgogne, Dijon, France.
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MeSH Terms
Descriptor/Qualifier:
Animals
Cells, Cultured
Hexanoic Acids / pharmacology*
Liver / drug effects*,  ultrastructure
Male
Microbodies / drug effects*
Molecular Conformation
Rats
Rats, Wistar
Structure-Activity Relationship
Chemical
Reg. No./Substance:
0/Hexanoic Acids

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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