Document Detail


Quantitation of combinatorial libraries of small organic molecules by normal-phase HPLC with evaporative light-scattering detection.
MedLine Citation:
PMID:  9237216     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
The advantages of evaporative light-scattering detection over UV detection for the quantitation of combinatorial libraries composed of small organic compounds by HPLC are described. The detector's response is independent of the sample chromophore, which makes it well-suited to chromatographic analyses of mixtures of dissimilar solutes. Thus, HPLC with evaporative light-scattering detection offers to potential for reducing false positive or false negative results in screening assays, because of its ability to detect the presence of impurities that absorb poorly in the UV (e.g., those impurities originating from the polymeric support). Furthermore, the evaporative light-scattering detector exhibits a nearly equivalent response to compounds of similar structural class. Hence, rapid quantitation of compound libraries may be carried out with the use of a single external standard. For example, the quantitation errors, based on a single external standard, for a series of steroids, hydantoins, and BOC- and Fmoc-protected amino acids by normal-phase HPLC with evaporative light-scattering detection average approximately +/-10%. The application of the evaporative light-scattering detector to the quantitation of low-level sample impurities and the detector's compatibility with gradient elution are also described.
Authors:
C E Kibbey
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Publication Detail:
Type:  Comparative Study; Journal Article    
Journal Detail:
Title:  Molecular diversity     Volume:  1     ISSN:  1381-1991     ISO Abbreviation:  Mol. Divers.     Publication Date:  1996 Aug 
Date Detail:
Created Date:  1997-09-23     Completed Date:  1997-09-23     Revised Date:  2006-11-15    
Medline Journal Info:
Nlm Unique ID:  9516534     Medline TA:  Mol Divers     Country:  NETHERLANDS    
Other Details:
Languages:  eng     Pagination:  247-58     Citation Subset:  IM    
Affiliation:
Parke-Davis Pharmaceutical Research, Division of Warner-Lambert Company, Ann Arbor, MI 48105, USA.
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MeSH Terms
Descriptor/Qualifier:
Amino Acids / chemistry
Chemistry, Organic / methods
Chromatography, High Pressure Liquid / methods*,  standards
Directed Molecular Evolution / methods*
Hydantoins / chemistry
Light
Reference Standards
Scattering, Radiation
Spectrophotometry, Ultraviolet
Steroids / chemistry,  standards
Chemical
Reg. No./Substance:
0/Amino Acids; 0/Hydantoins; 0/Steroids

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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