Document Detail


Protective effect of quercetin against intracerebral streptozotocin induced reduction in cerebral blood flow and impairment of memory in mice.
MedLine Citation:
PMID:  20096732     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
The aim of the present study is to investigate the effect of quercetin, a naturally occurring flavonoid, on cerebral blood flow (CBF), brain energy metabolism, memory impairment, oxidative stress and cholinergic dysfunction in brain following intracerebral (i.c.) streptozotocin (STZ) administration in mice. STZ (0.5mg/kg, i.c.) was administered twice at an interval of 48h. We found a significant reduction in CBF as measured by Laser Doppler Flowmetry (LDF). The brain energy metabolism was also altered as evidenced by significant reduction in brain ATP content. Daily treatment with quercetin (2.5, 5 and 10mg/kg, p.o.) starting from the first dose of STZ showed a dose-dependent restoration of CBF and ATP content. Further, quercetin prevented STZ induced memory impairment as assessed by Morris water maze and passive avoidance tests. Biochemical analysis revealed that STZ significantly increased malondialdehyde (MDA), nitrite and depleted glutathione (GSH) levels in the mice brain. Quercetin decreased oxidative and nitrosative stress as evidenced by a significant decrease in MDA, nitrite and increase in GSH levels. Quercetin also attenuated elevated acetylcholinesterase activity in the STZ-treated mice. Neither STZ (i.c.) nor quercetin showed any change in locomotor activity and blood glucose level. The present study demonstrates the beneficial effects of quercetin in improving CBF along with preventing memory impairment, oxidative stress, altered brain energy metabolism and cholinergic dysfunction caused by STZ in mice. Therefore, consumption of dietary stuff rich in quercetin should be encouraged to ward off dementia associated with vascular and neurodegenerative disorders.
Authors:
Santoshkumar Tota; Himani Awasthi; Pradeep Kumar Kamat; Chandishwar Nath; Kashif Hanif
Publication Detail:
Type:  Journal Article     Date:  2010-01-22
Journal Detail:
Title:  Behavioural brain research     Volume:  209     ISSN:  1872-7549     ISO Abbreviation:  Behav. Brain Res.     Publication Date:  2010 May 
Date Detail:
Created Date:  2010-03-03     Completed Date:  2010-05-25     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  8004872     Medline TA:  Behav Brain Res     Country:  Netherlands    
Other Details:
Languages:  eng     Pagination:  73-9     Citation Subset:  IM    
Affiliation:
Division of Pharmacology, Central Drug Research Institute, CSIR, Chattar Manzil, Lucknow, U.P., India.
Export Citation:
APA/MLA Format     Download EndNote     Download BibTex
MeSH Terms
Descriptor/Qualifier:
Acetylcholinesterase / metabolism
Adenosine Triphosphate / metabolism
Animals
Antibiotics, Antineoplastic / adverse effects,  pharmacology*
Antioxidants / pharmacology*
Avoidance Learning / drug effects
Blood Glucose / drug effects
Cerebrovascular Circulation / drug effects*
Dose-Response Relationship, Drug
Glutathione / metabolism
Injections, Intraventricular
Laser-Doppler Flowmetry / methods
Male
Malondialdehyde / metabolism
Maze Learning / drug effects
Memory Disorders / chemically induced*
Mice
Motor Activity / drug effects
Nitrites / metabolism
Quercetin / pharmacology*
Statistics, Nonparametric
Streptozocin / adverse effects,  pharmacology*
Chemical
Reg. No./Substance:
0/Antibiotics, Antineoplastic; 0/Antioxidants; 0/Blood Glucose; 0/Nitrites; 117-39-5/Quercetin; 18883-66-4/Streptozocin; 542-78-9/Malondialdehyde; 56-65-5/Adenosine Triphosphate; 70-18-8/Glutathione; EC 3.1.1.7/Acetylcholinesterase

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


Previous Document:  The chemotherapy agent, thioTEPA, yields long-term impairment of hippocampal cell proliferation and ...
Next Document:  Effects of single and simultaneous lesions of serotonergic and noradrenergic pathways on open-space ...