Document Detail


Phosphodiesterase-4 inhibition combined with isoniazid treatment of rabbits with pulmonary tuberculosis reduces macrophage activation and lung pathology.
MedLine Citation:
PMID:  21703411     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Tuberculosis (TB) is responsible for significant morbidity and mortality worldwide. Even after successful microbiological cure of TB, many patients are left with residual pulmonary damage that can lead to chronic respiratory impairment and greater risk of additional TB episodes due to reinfection with Mycobacterium tuberculosis. Elevated levels of the proinflammatory cytokine tumor necrosis factor-α and several other markers of inflammation, together with expression of matrix metalloproteinases, have been associated with increased risk of pulmonary fibrosis, tissue damage, and poor treatment outcomes in TB patients. In this study, we used a rabbit model of pulmonary TB to evaluate the impact of adjunctive immune modulation, using a phosphodiesterase-4 inhibitor that dampens the innate immune response, on the outcome of treatment with the antibiotic isoniazid. Our data show that cotreatment of M. tuberculosis infected rabbits with the phosphodiesterase-4 inhibitor CC-3052 plus isoniazid significantly reduced the extent of immune pathogenesis, compared with antibiotic alone, as determined by histologic analysis of infected tissues and the expression of genes involved in inflammation, fibrosis, and wound healing in the lungs. Combined treatment with an antibiotic and CC-3052 not only lessened disease but also improved bacterial clearance from the lungs. These findings support the potential for adjunctive immune modulation to improve the treatment of pulmonary TB and reduce the risk of chronic respiratory impairment.
Authors:
Selvakumar Subbian; Liana Tsenova; Paul O'Brien; Guibin Yang; Mi-Sun Koo; Blas Peixoto; Dorothy Fallows; Jerome B Zeldis; George Muller; Gilla Kaplan
Publication Detail:
Type:  Journal Article     Date:  2011-05-07
Journal Detail:
Title:  The American journal of pathology     Volume:  179     ISSN:  1525-2191     ISO Abbreviation:  Am. J. Pathol.     Publication Date:  2011 Jul 
Date Detail:
Created Date:  2011-06-27     Completed Date:  2011-10-28     Revised Date:  2012-02-15    
Medline Journal Info:
Nlm Unique ID:  0370502     Medline TA:  Am J Pathol     Country:  United States    
Other Details:
Languages:  eng     Pagination:  289-301     Citation Subset:  AIM; IM    
Copyright Information:
Copyright © 2011 American Society for Investigative Pathology. Published by Elsevier Inc. All rights reserved.
Affiliation:
Laboratory of Mycobacterial Immunity and Pathogenesis, The Public Health Research Institute at the University of Medicine and Dentistry of New Jersey, Newark, NJ 07103, USA.
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MeSH Terms
Descriptor/Qualifier:
Animals
Antitubercular Agents / therapeutic use*
Blotting, Western
Colony-Forming Units Assay
Cyclic Nucleotide Phosphodiesterases, Type 4 / chemistry*,  metabolism
Cytokines / metabolism
Drug Synergism
Drug Therapy, Combination
Female
Isoniazid / therapeutic use*
Lung / drug effects,  pathology*
Macrophage Activation / drug effects*
Male
Matrix Metalloproteinases / metabolism
Mycobacterium tuberculosis / pathogenicity
Phosphodiesterase 4 Inhibitors / therapeutic use
Pulmonary Fibrosis / enzymology,  pathology,  prevention & control
RNA, Messenger / genetics
Rabbits
Reverse Transcriptase Polymerase Chain Reaction
Thalidomide / analogs & derivatives*,  therapeutic use
Tuberculosis, Pulmonary / enzymology,  pathology,  prevention & control*
Grant Support
ID/Acronym/Agency:
R01 AI054338-11/AI/NIAID NIH HHS
Chemical
Reg. No./Substance:
0/Antitubercular Agents; 0/CC 3052; 0/Cytokines; 0/Phosphodiesterase 4 Inhibitors; 0/RNA, Messenger; 50-35-1/Thalidomide; 54-85-3/Isoniazid; EC 3.1.4.17/Cyclic Nucleotide Phosphodiesterases, Type 4; EC 3.4.24.-/Matrix Metalloproteinases

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