Document Detail


Pestalotiopsin a. Enantioselective construction of potential building blocks derived from antipodal cyclobutanol intermediates.
MedLine Citation:
PMID:  17696474     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
D-Glyceraldehyde acetonide has been used as the starting point for accessing the enantiomeric cyclobutanols 11 in optically pure condition. The dextrorotatory enantiomer has been transformed in five steps into the [3.2.0] bicyclic lactone 22. While the deoxygenation of 22 proved to be problematical, the uncyclized variant 25 underwent the Barton process smoothly. These findings guided the related conversion of (-)-11 into 34. Use was also made of ring-closing metathesis to bring about the conversion of (+)-11 into [4.2.0] bicyclic lactone building blocks. In general, all three pathways are efficient and offer the prospect of practical side-chain appendage for the purpose of installing the nine-membered ring of pestalotiopsin A (1).
Authors:
Leo A Paquette; Gregory D Parker; Takahiro Tei; Shuzhi Dong
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't     Date:  2007-08-15
Journal Detail:
Title:  The Journal of organic chemistry     Volume:  72     ISSN:  0022-3263     ISO Abbreviation:  J. Org. Chem.     Publication Date:  2007 Sep 
Date Detail:
Created Date:  2007-09-07     Completed Date:  2007-10-16     Revised Date:  2009-04-28    
Medline Journal Info:
Nlm Unique ID:  2985193R     Medline TA:  J Org Chem     Country:  United States    
Other Details:
Languages:  eng     Pagination:  7125-34     Citation Subset:  IM    
Affiliation:
Evans Chemical Laboratories, The Ohio State University, Columbus, OH 43210, USA. paquette.1@osu.edu
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MeSH Terms
Descriptor/Qualifier:
Alcohols / chemical synthesis*,  chemistry
Bicyclo Compounds / chemistry
Cyclobutanes / chemical synthesis*,  chemistry
Lactones / chemistry
Sesquiterpenes / chemical synthesis*
Stereoisomerism
Chemical
Reg. No./Substance:
0/Alcohols; 0/Bicyclo Compounds; 0/Cyclobutanes; 0/Lactones; 0/Sesquiterpenes; 0/pestalotiopsin A
Comments/Corrections
Erratum In:
J Org Chem. 2009 Feb 20;74(4):1812

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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