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Parallel supported synthesis of polyamine-imidazole conjugates.
MedLine Citation:
PMID:  15575667     Owner:  NLM     Status:  PubMed-not-MEDLINE    
Abstract/OtherAbstract:
[reaction: see text] A small collection of nine polyamine-imidazole conjugates, potentially acting as RNases A mimics, has been synthesized on SynPhase lanterns using amino alcohols and diamines as building blocks. Couplings were performed via S(N)2 alkylation of methanesulfonates with amines. The final introduction of N-4-nitrobenzyloxycarbonyldiamines allowed easy purification of the cleaved compounds.
Authors:
Sylvie Picard; Myriam Le Roch; Jacques Renault; Philippe Uriac
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Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Organic letters     Volume:  6     ISSN:  1523-7060     ISO Abbreviation:  Org. Lett.     Publication Date:  2004 Dec 
Date Detail:
Created Date:  2004-12-03     Completed Date:  2005-05-17     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  100890393     Medline TA:  Org Lett     Country:  United States    
Other Details:
Languages:  eng     Pagination:  4711-4     Citation Subset:  -    
Affiliation:
Université Rennes 1, Institut de Chimie de Rennes, Synthèse et Extraction de Molécules à Visée Thérapeutique, Faculté des Sciences Biologiques et Médicales, 2 avenue du professeur Léon Bernard, 35043 Rennes, France.
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