Document Detail


Nitrosation of aryl and heteroaryltrifluoroborates with nitrosonium tetrafluoroborate.
MedLine Citation:
PMID:  22524190     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Organotrifluoroborates have emerged as an alternative to toxic and air- and moisture-sensitive organometallic species for the synthesis of functionalized aryl and heteroaryl compounds. It has been shown that the trifluoroborate moiety can be easily converted into a variety of different substituents in a late synthetic stage. In this paper, we disclose a mild, selective, and convenient method for the ipso-nitrosation of organotrifluoroborates using nitrosonium tetrafluoroborate (NOBF(4)). Aryl- and heteroaryltrifluoroborates were converted into the corresponding nitroso products in good to excellent yields. This method proved to be tolerant of a broad range of functional groups.
Authors:
Gary A Molander; Livia N Cavalcanti
Publication Detail:
Type:  Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't     Date:  2012-04-24
Journal Detail:
Title:  The Journal of organic chemistry     Volume:  77     ISSN:  1520-6904     ISO Abbreviation:  J. Org. Chem.     Publication Date:  2012 May 
Date Detail:
Created Date:  2012-05-04     Completed Date:  2012-09-28     Revised Date:  2013-05-06    
Medline Journal Info:
Nlm Unique ID:  2985193R     Medline TA:  J Org Chem     Country:  United States    
Other Details:
Languages:  eng     Pagination:  4402-13     Citation Subset:  IM    
Affiliation:
Roy and Diana Vagelos Laboratories, Department of Chemistry, University of Pennsylvania, 231 South 34th Street, Philadelphia, Pennsylvania 19104-6323, USA. gmolandr@sas.upenn.edu
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MeSH Terms
Descriptor/Qualifier:
Borates / chemical synthesis,  chemistry*
Catalysis
Heterocyclic Compounds / chemistry*
Molecular Structure
Nitric Oxide / chemical synthesis*,  chemistry*
Nitrosation
Grant Support
ID/Acronym/Agency:
GM035249/GM/NIGMS NIH HHS; R01 GM035249/GM/NIGMS NIH HHS; R01 GM081376/GM/NIGMS NIH HHS; R01 GM086209/GM/NIGMS NIH HHS; S10 RR016640/RR/NCRR NIH HHS
Chemical
Reg. No./Substance:
0/Borates; 0/Heterocyclic Compounds; 10102-43-9/Nitric Oxide; 14635-75-7/nitrosonium tetrafluoroborate

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