Document Detail


Neuroprotection by excitatory amino acid antagonist augments the benefit of thrombolysis in embolic stroke in rats.
MedLine Citation:
PMID:  8236347     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
BACKGROUND AND PURPOSE: The effects of delayed thrombolysis with alteplase and neuroprotection with an excitatory amino acid receptor antagonist and their combination were tested in an embolic stroke model. METHODS: In 61 rats the carotid artery territory was embolized with arterial-like fibrin-rich clots. Hemispheric cerebral blood flow before and after embolization was measured by intra-arterial 133Xe injection method. The animals were assigned to one of the following treatments: (1) vehicle-treated controls (n = 15); (2) dizocilpine 1 mg/kg i.v. 5 minutes after embolization (n = 16); (3) alteplase 20 mg/kg as an intravenous continuous infusion starting 2 hours after embolization (n = 16); and (4) both agents (n = 14). Carotid angiography displayed the site of occlusion of the cerebral arterial tree immediately after and 3 hours after embolization, and the clinical neurological score was assessed after the rats recovered from anesthesia and before the rats were killed. Brains were fixed after 2 days and evaluated neuropathologically; infarct volume affecting cortical and deep brain structures was measured separately. RESULTS: Both alteplase and dizocilpine reduced the total infarct volume (P = .05 and P = .04, respectively, Mann-Whitney tests). Dizocilpine reduced the incidence of cortical infarctions by 48% (P < .001, Fisher's test). Only the combined treatment significantly reduced deep brain infarctions (P = .03, Mann-Whitney test). The combined treatment also improved the clinical score by 83% compared with controls, by 75% compared with the group treated by dizocilpine alone, and by 50% compared with the group treated by alteplase alone. Sixty-seven percent of thrombolytic-treated animals recanalized completely compared with 39% of those given no thrombolytics (P = .05, Fisher's test). The clinical outcome correlated with infarct size (P < .01, Spearman test). CONCLUSIONS: Our results document comparable efficacy of delayed thrombolysis and excitatory amino acid receptor antagonism in this model and suggest that combination of these two therapeutic approaches may yield additional benefit in treatment of thromboembolic stroke, particularly in cases where deep brain (end-artery-supplied) structures are affected.
Authors:
T Sereghy; K Overgaard; G Boysen
Related Documents :
12739237 - Targeting of post-ischemic cerebral endothelium in rat by liposomes bearing polyethylen...
11341477 - Effects of dexmedetomidine after transient and permanent occlusion of the middle cerebr...
9221957 - Expressions of p-selectin- and hsp72-like immunoreactivities in rat brain after transie...
20041427 - Cornin ameliorates cerebral infarction in rats by antioxidant action and stabilization ...
4330087 - Regulation of gluconeogenesis during exposure of young rats to hypoxic conditions.
2505007 - Striatal dopamine, sexual activity and lifespan. longevity of rats treated with (-)depr...
Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Stroke; a journal of cerebral circulation     Volume:  24     ISSN:  0039-2499     ISO Abbreviation:  Stroke     Publication Date:  1993 Nov 
Date Detail:
Created Date:  1993-11-29     Completed Date:  1993-11-29     Revised Date:  2003-11-14    
Medline Journal Info:
Nlm Unique ID:  0235266     Medline TA:  Stroke     Country:  UNITED STATES    
Other Details:
Languages:  eng     Pagination:  1702-8     Citation Subset:  IM    
Affiliation:
Department of Neurology, University Hospital of Copenhagen, Rigshospitalet, Denmark.
Export Citation:
APA/MLA Format     Download EndNote     Download BibTex
MeSH Terms
Descriptor/Qualifier:
Animals
Blood Pressure / drug effects
Brain / pathology*
Carbon Dioxide / blood
Cerebral Angiography
Cerebral Infarction / pathology,  physiopathology,  prevention & control*
Dizocilpine Maleate / therapeutic use*
Drug Therapy, Combination
Infusions, Intravenous
Intracranial Embolism and Thrombosis / drug therapy*,  pathology,  physiopathology
Male
N-Methylaspartate / antagonists & inhibitors
Oxygen / blood
Partial Pressure
Rats
Rats, Sprague-Dawley
Thrombolytic Therapy*
Time Factors
Tissue Plasminogen Activator / administration & dosage,  therapeutic use*
Chemical
Reg. No./Substance:
124-38-9/Carbon Dioxide; 6384-92-5/N-Methylaspartate; 77086-22-7/Dizocilpine Maleate; 7782-44-7/Oxygen; EC 3.4.21.68/Tissue Plasminogen Activator
Comments/Corrections
Erratum In:
Stroke 1997 Feb;28(2):466

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


Previous Document:  Cerebellar infarction. Clinical and neuroimaging analysis in 293 patients. The Tohoku Cerebellar Inf...
Next Document:  Improved posthypoxic recovery of synaptic transmission in gerbil neocortical slices treated with a c...