Document Detail


NMDA receptor-nitric oxide transmission mediates neuronal iron homeostasis via the GTPase Dexras1.
MedLine Citation:
PMID:  16908409     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Dexras1 is a 30 kDa G protein in the Ras subfamily whose discovery was based on its pronounced inducibility by the glucocorticoid dexamethasone. It binds to neuronal nitric oxide synthase (nNOS) via the adaptor protein CAPON, eliciting S-nitrosylation and activation of Dexras1. We report that Dexras1 binds to the peripheral benzodiazepine receptor-associated protein (PAP7), a protein of unknown function that binds to cyclic AMP-dependent protein kinase and the peripheral benzodiazepine receptor. PAP7 in turn binds to the divalent metal transporter (DMT1), an iron import channel. We have identified a signaling cascade in neurons whereby stimulation of NMDA receptors activates nNOS, leading to S-nitrosylation and activation of Dexras1, which, via PAP7 and DMT1, physiologically induces iron uptake. As selective iron chelation prevents NMDA neurotoxicity in cortical cultures, the NMDA-NO-Dexras1-PAP7-DMT1-iron uptake signaling cascade also appears to mediate NMDA neurotoxicity.
Authors:
Jaime H Cheah; Sangwon F Kim; Lynda D Hester; Kathleen W Clancy; Stanley E Patterson; Vassilios Papadopoulos; Solomon H Snyder
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Publication Detail:
Type:  Comparative Study; Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  Neuron     Volume:  51     ISSN:  0896-6273     ISO Abbreviation:  Neuron     Publication Date:  2006 Aug 
Date Detail:
Created Date:  2006-08-15     Completed Date:  2006-09-26     Revised Date:  2011-08-25    
Medline Journal Info:
Nlm Unique ID:  8809320     Medline TA:  Neuron     Country:  United States    
Other Details:
Languages:  eng     Pagination:  431-40     Citation Subset:  IM    
Affiliation:
Department of Neuroscience, Johns Hopkins University School of Medicine, Baltimore, Maryland 21205, USA.
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MeSH Terms
Descriptor/Qualifier:
Adaptor Proteins, Signal Transducing
Aldehydes / pharmacology
Animals
Blotting, Western / methods
Cation Transport Proteins / metabolism
Cells, Cultured
Cerebral Cortex / cytology
Dizocilpine Maleate / pharmacology
Dose-Response Relationship, Drug
Drug Interactions
Embryo, Mammalian
Excitatory Amino Acid Agents / pharmacology
Fluorescent Antibody Technique / methods
Homeostasis / drug effects,  physiology*
Humans
Hydrazones / pharmacology
Immunoprecipitation / methods
Iron / metabolism*
Iron Chelating Agents / pharmacology
Iron-Binding Proteins / metabolism
Membrane Proteins
Mice
Mice, Knockout
Models, Biological
N-Methylaspartate / pharmacology
Neurons / drug effects,  metabolism
Nitric Oxide / physiology*
Nitric Oxide Synthase Type I / deficiency,  metabolism
Protein Binding / drug effects,  physiology
Rats
Reactive Oxygen Species / immunology,  metabolism
Receptors, GABA-A / metabolism
Receptors, N-Methyl-D-Aspartate / physiology*
Signal Transduction / drug effects,  physiology*
Transfection / methods
ras Proteins / physiology*
Grant Support
ID/Acronym/Agency:
DA000266/DA/NIDA NIH HHS; DA00074/DA/NIDA NIH HHS; K99 MH079614-01/MH/NIMH NIH HHS
Chemical
Reg. No./Substance:
0/Acbd3 protein, mouse; 0/Adaptor Proteins, Signal Transducing; 0/Aldehydes; 0/Cation Transport Proteins; 0/Excitatory Amino Acid Agents; 0/Hydrazones; 0/Iron Chelating Agents; 0/Iron-Binding Proteins; 0/Membrane Proteins; 0/Reactive Oxygen Species; 0/Receptors, GABA-A; 0/Receptors, N-Methyl-D-Aspartate; 0/salicylaldehyde isonicotinoyl hydrazone; 0/solute carrier family 11- (proton-coupled divalent metal ion transporters), member 2; 10102-43-9/Nitric Oxide; 6384-92-5/N-Methylaspartate; 7439-89-6/Iron; 77086-22-7/Dizocilpine Maleate; EC 1.14.13.39/Nitric Oxide Synthase Type I; EC 3.6.1.-/Rasd1 protein, mouse; EC 3.6.5.2/ras Proteins
Comments/Corrections

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