Document Detail


N-benzyl aspartate nitrones: unprecedented single-step synthesis and [3 + 2] cycloaddition reactions with alkenes.
MedLine Citation:
PMID:  18785749     Owner:  NLM     Status:  PubMed-not-MEDLINE    
Abstract/OtherAbstract:
N-benzyl aspartate nitrones 2, prepared by addition of N-benzylhydroxylamine to dialkyl acetylenedicarboxylates 1, underwent [3 + 2] thermal cycloaddition with a wide range of alkenes to afford isoxazolidines 4 bearing a polyfunctionalized quaternary center. Under these uncatalyzed conditions, the trans stereocontrol observed with vinyl ethers is higher than that obtained with all acyclic activated nitrones reported to date. The first asymmetric access to a type-4 pure adduct was achieved starting from the chiral aspartate nitrone derived from (S)-alpha-methylbenzylhydroxylamine.
Authors:
Thanh Binh Nguyen; Arnaud Martel; Robert Dhal; Gilles Dujardin
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Publication Detail:
Type:  Journal Article     Date:  2008-09-12
Journal Detail:
Title:  Organic letters     Volume:  10     ISSN:  1523-7052     ISO Abbreviation:  Org. Lett.     Publication Date:  2008 Oct 
Date Detail:
Created Date:  2008-10-09     Completed Date:  2008-12-10     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  100890393     Medline TA:  Org Lett     Country:  United States    
Other Details:
Languages:  eng     Pagination:  4493-6     Citation Subset:  -    
Affiliation:
UCO2M UMR 6011 & IRIM2F FR 2575 CNRS, Université du Maine, 72085, Le Mans, France.
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