Document Detail


N-acetylphytosphingosine enhances the radiosensitivity of lung cancer cell line NCI-H460.
MedLine Citation:
PMID:  18414010     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Ceramides are well-known second messengers that induce apoptosis in various kinds of cancer cells, and their effects are closely related to radiation sensitivity. Phytoceramides, the yeast counterparts of the mammalian ceramides, are also reported to induce apoptosis. We investigated the effect of a novel ceramide derivative, N-acetylphytosphingosine (NAPS), on the radiosensitivity of NCI-H460 human lung carcinoma cells and its differential cytotoxicity in tumor and normal cells. The combination of NAPS with radiation significantly increased clonogenic cell death and caspase-dependent apoptosis. The combined treatment greatly increased Bax expression and Bid cleavage, but not Bcl-2 expression. However, there was no effect on radiosensitivity and apoptosis in BEAS2B cells, which derive from normal human bronchial epithelium. Cell proliferation and DNA synthesis were significantly inhibited by NAPS in both NCI-H460 and BEAS2B cells, but only the BEAS2B cells recovered by 48h after removal of the NAPS. Furthermore, the NCI-H460 cells underwent more DNA fragmentation than the BEAS2B cells in response to NAPS. Our results indicate that NAPS may be a potential radiosensitizing agent with differential effects on tumor vs. normal cells.
Authors:
Youngsoo Han; Kisung Kim; Ji-Young Shim; Changsoe Park; Jie-Young Song; Yeon-Sook Yun
Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't     Date:  2008-03-31
Journal Detail:
Title:  Molecules and cells     Volume:  25     ISSN:  1016-8478     ISO Abbreviation:  Mol. Cells     Publication Date:  2008 Apr 
Date Detail:
Created Date:  2008-05-27     Completed Date:  2008-08-04     Revised Date:  2009-03-12    
Medline Journal Info:
Nlm Unique ID:  9610936     Medline TA:  Mol Cells     Country:  Korea (South)    
Other Details:
Languages:  eng     Pagination:  224-30     Citation Subset:  IM    
Affiliation:
Laboratory of Radiation Sensitization and Protection, Korea Institute of Radiological and Medical Sciences, Seoul 139-706, Korea.
Export Citation:
APA/MLA Format     Download EndNote     Download BibTex
MeSH Terms
Descriptor/Qualifier:
Caspases / metabolism
Cell Death / drug effects,  radiation effects
Cell Line, Tumor
Cell Survival / drug effects,  radiation effects
Clone Cells
Cytostatic Agents / pharmacology
Enzyme Activation / drug effects,  radiation effects
Gamma Rays
Humans
Lung Neoplasms / enzymology,  pathology*
Radiation Tolerance / drug effects*
Sphingolipids / pharmacology*
bcl-2-Associated X Protein / metabolism
Chemical
Reg. No./Substance:
0/Cytostatic Agents; 0/N-acetylphytosphingosine; 0/Sphingolipids; 0/bcl-2-Associated X Protein; EC 3.4.22.-/Caspases
Comments/Corrections
Erratum In:
Mol Cells. 2009 Jan;27(1):125

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


Previous Document:  Expressed sequence tag analysis of Antarctic hairgrass Deschampsia antarctica from King George Islan...
Next Document:  Development of a sequence characteristic amplified region marker linked to the L4 locus conferring b...