Document Detail


Mefloquine tolerability during chemoprophylaxis: focus on adverse event assessments, stereochemistry and compliance.
MedLine Citation:
PMID:  8765456     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
This longitudinal study of travellers to Africa taking mefloquine (MQ) chemoprophylaxis aimed to quantify and assess non-serious adverse events (AE) occurring during short-term prophylaxis and relate these to concentrations of racemic MQ, its enantiomers and metabolite. A total of 420 volunteers (52% F) participated. AEs with some impact on activities were reported by 11.2% of participants including 7.9% of neurological/psychiatric symptoms. Women were more likely to report AEs (P = 0.02). The standardized questionnaires used showed more pathological indicators in travellers who reported subjective AE with significantly more dizziness, distress, sleep disturbances and a high total mood disturbance (TMD) in the AE group. There was, however, no significant performance deficit in computerized psychomotor tests in those experiencing AE. Furthermore, no significant differences were observed in enantiomer ratios, metabolite concentrations, or racemic MQ levels in participants with or without AEs suggesting that these factors are not the main predictors of mefloquine intolerability.
Authors:
P Schlagenhauf; R Steffen; H Lobel; R Johnson; R Letz; A Tschopp; N Vranjes; Y Bergqvist; O Ericsson; U Hellgren; L Rombo; S Mannino; J Handschin; D Stürchler
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  Tropical medicine & international health : TM & IH     Volume:  1     ISSN:  1360-2276     ISO Abbreviation:  Trop. Med. Int. Health     Publication Date:  1996 Aug 
Date Detail:
Created Date:  1996-09-13     Completed Date:  1996-09-13     Revised Date:  2006-11-15    
Medline Journal Info:
Nlm Unique ID:  9610576     Medline TA:  Trop Med Int Health     Country:  ENGLAND    
Other Details:
Languages:  eng     Pagination:  485-94     Citation Subset:  IM    
Affiliation:
Institute for Social and Preventive Medicine, University of Zürich.
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MeSH Terms
Descriptor/Qualifier:
Adolescent
Adult
Africa
Drug Tolerance
Female
Humans
Longitudinal Studies
Malaria, Falciparum / prevention & control*
Male
Mefloquine / adverse effects*,  chemistry
Middle Aged
Patient Compliance
Questionnaires
Sex Factors
Stereoisomerism
Travel
Chemical
Reg. No./Substance:
53230-10-7/Mefloquine

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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