Document Detail


Mechanisms involved in ceramide-induced cell cycle arrest in human hepatocarcinoma cells.
MedLine Citation:
PMID:  17373752     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
AIM: To investigate the effect of ceramide on the cell cycle in human hepatocarcinoma Bel7402 cells. Possible molecular mechanisms were explored. METHODS: [3- (4, 5)-dimethylthiazol-2-yl]-2, 5-diphenyltetrazolium bromide (MTT) assay, plasmid transfection, reporter assay, FACS and Western blotting analyses were employed to investigate the effect and the related molecular mechanisms of C2-ceramide on the cell cycle of Bel7402 cells. RESULTS: C2-ceramide was found to inhibit the growth of Bel7402 cells by inducing cell cycle arrest. During the process, the expression of p21 protein increased, while that of cyclinD1, phospho-ERK1/2 and c-myc decreased. Furthermore, the level of CDK7 was downregulated, while the transcriptional activity of PPARgamma was upregulated. Addition of GW9662, which is a PPARgamma specific antagonist, could reserve the modulation action on CDK7. CONCLUSION: Our results support the hypothesis that cell cycle arrest induced by C2-ceramide may be mediated via accumulation of p21 and reduction of cyclinD1 and CDK7, at least partly, through PPARgamma activation. The ERK signaling pathway was involved in this process.
Authors:
Jing Wang; Xiao-Wen Lv; Jie-Ping Shi; Xiao-Song Hu
Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  World journal of gastroenterology : WJG     Volume:  13     ISSN:  1007-9327     ISO Abbreviation:  World J. Gastroenterol.     Publication Date:  2007 Feb 
Date Detail:
Created Date:  2007-03-21     Completed Date:  2007-06-06     Revised Date:  2009-11-19    
Medline Journal Info:
Nlm Unique ID:  100883448     Medline TA:  World J Gastroenterol     Country:  China    
Other Details:
Languages:  eng     Pagination:  1129-34     Citation Subset:  IM    
Affiliation:
Research Center for Eco-Environmental Sciences, The Chinese Academy of Sciences, Haidian District, Beijing 100085, China. wangjing@rcees.ac.cn
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MeSH Terms
Descriptor/Qualifier:
Carcinoma, Hepatocellular / metabolism*,  pathology
Cell Cycle / drug effects*,  physiology
Cell Line, Tumor
Cell Proliferation / drug effects
Cyclin D1 / genetics,  metabolism
Cyclin-Dependent Kinase Inhibitor p21 / genetics,  metabolism
Cyclin-Dependent Kinases / genetics,  metabolism
Enzyme Inhibitors / pharmacology*
Extracellular Signal-Regulated MAP Kinases / physiology
Gene Expression Regulation / drug effects
Humans
Liver Neoplasms / metabolism*,  pathology
PPAR gamma / physiology
Signal Transduction / physiology
Sphingosine / analogs & derivatives*,  pharmacology
Chemical
Reg. No./Substance:
0/Cyclin-Dependent Kinase Inhibitor p21; 0/Enzyme Inhibitors; 0/N-acetylsphingosine; 0/PPAR gamma; 123-78-4/Sphingosine; 136601-57-5/Cyclin D1; EC 2.7.1.37/cyclin-dependent kinase-activating kinase; EC 2.7.11.22/Cyclin-Dependent Kinases; EC 2.7.11.24/Extracellular Signal-Regulated MAP Kinases

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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