Document Detail


Kidney and liver contributions to salicylate metabolism in rats.
MedLine Citation:
PMID:  7957447     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
The pharmacokinetics and metabolism of radiolabelled salicylate were studied in rats and compared with that of the isolated perfused rat liver and the perfused rat kidney. Both parent compound and salicylate metabolites (mainly conjugates with glycine and glucuronic acid) were eliminated mostly into urine. The comparison of a relative proportion of metabolites eliminated in whole rats with that of the isolated perfused rat liver and the perfused rat kidney showed that both kidney and liver contributed to the salicylate metabolism. The glycine conjugate of salicylate was formed predominantly in the kidney whereas both kidney and liver participated in the formation of glucuronic acid derivatives.
Authors:
M Láznícek; A Láznícková
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Publication Detail:
Type:  In Vitro; Journal Article    
Journal Detail:
Title:  European journal of drug metabolism and pharmacokinetics     Volume:  19     ISSN:  0378-7966     ISO Abbreviation:  Eur J Drug Metab Pharmacokinet     Publication Date:    1994 Jan-Mar
Date Detail:
Created Date:  1994-12-07     Completed Date:  1994-12-07     Revised Date:  2011-02-02    
Medline Journal Info:
Nlm Unique ID:  7608491     Medline TA:  Eur J Drug Metab Pharmacokinet     Country:  SWITZERLAND    
Other Details:
Languages:  eng     Pagination:  21-6     Citation Subset:  IM    
Affiliation:
Faculty of Pharmacy, Charles University, Hradec Králové, Czechoslovakia.
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MeSH Terms
Descriptor/Qualifier:
Animals
Biotransformation
Gluconates / metabolism,  urine
Glycine / metabolism,  urine
Half-Life
Kidney / metabolism*
Liver / metabolism*
Male
Rats
Rats, Wistar
Salicylic Acid
Salicylic Acids / pharmacokinetics*,  urine
Technetium Tc 99m Pentetate
Tissue Distribution
Chemical
Reg. No./Substance:
0/Gluconates; 0/Salicylic Acids; 56-40-6/Glycine; 65454-61-7/Technetium Tc 99m Pentetate; 69-72-7/Salicylic Acid

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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