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Inhibition of urease by extracts derived from 15 Chinese medicinal herbs.
MedLine Citation:
PMID:  21639688     Owner:  NLM     Status:  In-Data-Review    
Abstract/OtherAbstract:
Context: Helicobacter pylori is a major causative factor in gastritis-like disorders, and urease plays a key role in Helicobacter pylori colonizing and persisting in the mucous layer of the human stomach. In China, a variety of Chinese medicinal herbs have been prescribed to attenuate or eradicate gastritis-like disorders. However, little is known about the urease inhibition of Chinese medicinal herbs. Objective: The present study was conducted to investigate the urease inhibition activities of the ethanol and water extracts of 15 Chinese medicinal herbs. Materials and methods: The ethanol and water extracts derived from 15 medicinal herbs, traditionally used for the treatment of gastritis-like disorders in China, were tested for urease-inhibition activity using the phenol red method. Results: Screened at 10 µg/mL, 14 ethanol extracts and 10 water extracts showed urease inhibition. The ethanol extracts of Magnolia officinalis Rehd. et Wils. (Magnoliaceae) and Cassia obtusifolia L. (Leguminosae) possessed inhibition rates higher than 50% with IC(50) values of 6.5 and 12.3 µg/mL, respectively. After fractionating successively, the petroleum ether fraction of the ethanol extracts of Magnolia officinalis showed the best activity with 90.8% urease inhibition at a concentration of 10 µg/mL. The bioautography of the petroleum ether fraction indicated the existence of the urease inhibitors in the herb. Discussion and conclusion: The present results indicated that some Chinese medicinal herbs might treat gastritis-like disorders via the inhibition of Helicobacter pylori urease and the further possibility for discovering useful novel urease inhibitors from the Chinese medicinal herbs.
Authors:
Da-Hua Shi; Yu-Wei Liu; Wei-Wei Liu; Zhi-Feng Gu
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Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Pharmaceutical biology     Volume:  49     ISSN:  1744-5116     ISO Abbreviation:  Pharm Biol     Publication Date:  2011 Jul 
Date Detail:
Created Date:  2011-06-06     Completed Date:  -     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  9812552     Medline TA:  Pharm Biol     Country:  England    
Other Details:
Languages:  eng     Pagination:  752-5     Citation Subset:  IM    
Affiliation:
School of Chemical Engineering, Huaihai Institute of Technology, Lianyungang, People's Republic of China.
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