Document Detail


Informatics, machine learning and computational medicinal chemistry.
MedLine Citation:
PMID:  21452981     Owner:  NLM     Status:  In-Data-Review    
Abstract/OtherAbstract:
This article reviews the use of informatics and computational chemistry methods in medicinal chemistry, with special consideration of how computational techniques can be adapted and extended to obtain more and higher-quality information. Special consideration is given to the computation of protein-ligand binding affinities, to the prediction of off-target bioactivities, bioactivity spectra and computational toxicology, and also to calculating absorption-, distribution-, metabolism- and excretion-relevant properties, such as solubility.
Authors:
John Bo Mitchell
Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  Future medicinal chemistry     Volume:  3     ISSN:  1756-8927     ISO Abbreviation:  Future Med Chem     Publication Date:  2011 Mar 
Date Detail:
Created Date:  2011-04-01     Completed Date:  -     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  101511162     Medline TA:  Future Med Chem     Country:  England    
Other Details:
Languages:  eng     Pagination:  451-67     Citation Subset:  IM    
Affiliation:
Centre for Biomolecular Sciences, University of St Andrews, North Haugh, St Andrews KY16 9ST, UK. jbom@st-andrews.ac.uk.
Export Citation:
APA/MLA Format     Download EndNote     Download BibTex
MeSH Terms
Descriptor/Qualifier:

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


Previous Document:  Novel neuraminidase inhibitors: identification, biological evaluation and investigations of the bind...
Next Document:  What has polar surface area ever done for drug discovery?