Document Detail


Identification of a monopartite sequence in PU.1 essential for nuclear import, DNA-binding and transcription of myeloid-specific genes.
MedLine Citation:
PMID:  17340619     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
The Ets transcription factor PU.1 is an essential regulator of normal hematopoiesis, especially within the myeloid lineage. As such, endogenous PU.1 predominantly localizes to the nucleus of mammalian cells to facilitate gene regulation. However, to date, little is known regarding the mechanisms of PU.1 nuclear transport. We found, using HeLa and RAW 264.7 macrophage cells, that PU.1 enters the nucleus via passive diffusion and active transport. The latter can be facilitated by: (i) the classical pathway requiring importin alpha and beta; (ii) the non-classical pathway requiring only importin beta; or (iii) direct interaction with nucleoporins. A group of six positively charged lysine or arginine residues within the Ets DNA-binding domain was determined to be crucial in active nuclear import. These residues directly interact with importin beta to facilitate a predominantly non-classical import pathway. Furthermore, luciferase reporter assays demonstrated that these same six amino acids are crucial for PU.1-mediated transcriptional activation of myeloid-specific genes. Indeed, these residues may represent a consensus sequence vital for nuclear import, DNA-binding and transcriptional activity of Ets family members. By identifying and characterizing the mechanisms of PU.1 nuclear import and the specific amino acids involved, this report may provide insights into the molecular basis of diseases.
Authors:
Juliana C Kwok; José Perdomo; Beng H Chong
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  Journal of cellular biochemistry     Volume:  101     ISSN:  0730-2312     ISO Abbreviation:  J. Cell. Biochem.     Publication Date:  2007 Aug 
Date Detail:
Created Date:  2007-07-31     Completed Date:  2008-04-09     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  8205768     Medline TA:  J Cell Biochem     Country:  United States    
Other Details:
Languages:  eng     Pagination:  1456-74     Citation Subset:  IM    
Affiliation:
Centre for Thrombosis and Vascular Research, Department of Medicine, St. George Clinical School, University of New South Wales, Sydney, New South Wales, Australia. j.kwok@unsw.edu.au
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MeSH Terms
Descriptor/Qualifier:
Active Transport, Cell Nucleus / physiology*
Amino Acid Sequence*
Animals
Cell Nucleus / metabolism
Cells, Cultured
DNA / metabolism*
Gene Expression Regulation
Genes, Reporter
Hela Cells
Humans
Macrophages / cytology,  metabolism
Mice
Models, Molecular
Molecular Sequence Data
Mutation
Protein Binding
Protein Structure, Tertiary
Proto-Oncogene Proteins / chemistry,  genetics*,  metabolism*
Recombinant Fusion Proteins / genetics,  metabolism
Sequence Alignment
Trans-Activators / chemistry,  genetics*,  metabolism*
Transcription, Genetic*
Chemical
Reg. No./Substance:
0/Proto-Oncogene Proteins; 0/Recombinant Fusion Proteins; 0/Trans-Activators; 0/proto-oncogene protein Spi-1; 9007-49-2/DNA

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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