Document Detail


Expression of kinin B1 receptors in the spinal cord of streptozotocin-diabetic rat.
MedLine Citation:
PMID:  15538175     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Previous studies have reported cardiovascular and nociceptive responses after intrathecal injection of kinin B1 receptor (B1R) agonists in the model of streptozotocin (STZ)-diabetic rat (diabetic). The aim of this study was to measure the early up-regulation of B1R binding sites and mRNA in the thoracic spinal cord of diabetic and control rats. Data show significant increases of specific B1R binding sites in the dorsal horn of diabetic rats 2 days (+315%), 7 days (+303%) and 21 days (+181%) after STZ treatment. Levels of mRNA were significantly increased (+68%) at 2 and 7 days but not at 21 days. These data bring the first molecular evidence for an early up-regulation of B1R in the spinal cord of diabetic rat.
Authors:
Brice Ongali; Maria Martha Campos; Mihai Petcu; Donata Rodi; Frank Cloutier; Jean-Guy Chabot; Gaétan Thibault; Réjean Couture
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Publication Detail:
Type:  Comparative Study; Journal Article; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  Neuroreport     Volume:  15     ISSN:  0959-4965     ISO Abbreviation:  Neuroreport     Publication Date:  2004 Nov 
Date Detail:
Created Date:  2004-11-11     Completed Date:  2005-03-14     Revised Date:  2006-11-15    
Medline Journal Info:
Nlm Unique ID:  9100935     Medline TA:  Neuroreport     Country:  England    
Other Details:
Languages:  eng     Pagination:  2463-6     Citation Subset:  IM    
Affiliation:
Department of Physiology, Université de Montréal, Pavillon Paul-G.-Desmarais, 2960, Chemin de la Tour, Montréal, Québec, H3T 1J4, Canada.
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MeSH Terms
Descriptor/Qualifier:
Animals
Blood Glucose / metabolism
Body Weight / physiology
Bradykinin / analogs & derivatives*,  pharmacokinetics
Diabetes Mellitus, Experimental / metabolism*
Gene Expression Regulation / drug effects
In Situ Hybridization / methods
Iodine Isotopes / pharmacokinetics
Male
Protein Binding / drug effects,  physiology
RNA, Messenger / metabolism
Radiography / methods
Rats
Rats, Wistar
Receptor, Bradykinin B1 / genetics,  metabolism*
Reverse Transcriptase Polymerase Chain Reaction / methods
Spinal Cord / metabolism*
Tetrahydroisoquinolines / pharmacokinetics
Time Factors
Chemical
Reg. No./Substance:
0/Blood Glucose; 0/Iodine Isotopes; 0/RNA, Messenger; 0/Receptor, Bradykinin B1; 0/Tetrahydroisoquinolines; 138680-92-9/HOE 140, desArg(10)-; 58-82-2/Bradykinin

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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