Document Detail


Effects of CP-060S, a novel cardioprotective drug, on cardiac function and myocardial oxygen consumption.
MedLine Citation:
PMID:  9888255     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
1. We examined the effects of CP-060S on cardiac function and myocardial oxygen consumption (MVO2) in anesthetized dogs. 2. CP-060S (10-300 microg/kg i.v.) decreased heart rate, increased aortic flow and decreased mean blood pressure in a dose-dependent manner. The PR interval was significantly prolonged by administration of CP-060S (300 microg/kg i.v.). 3. CP-060S (10-300 microg/kg i.v.) increased coronary blood flow in a dose-dependent manner. Left ventricular end-diastolic pressure and maximal first derivative of left ventricular pressure were not significantly affected. 4. CP-060S (10-300 microg/kg i.v.) increased coronary sinus blood flow and decreased arteriovenous oxygen difference and MVO2 in a dose-dependent manner. 5. The effects of CP-060S on cardiac function and MVO2 are qualitatively similar to those of diltiazem, a typical Ca2+ antagonist.
Authors:
Y Suzuki; M Akima; K Tamura
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Publication Detail:
Type:  Journal Article    
Journal Detail:
Title:  General pharmacology     Volume:  32     ISSN:  0306-3623     ISO Abbreviation:  Gen. Pharmacol.     Publication Date:  1999 Jan 
Date Detail:
Created Date:  1999-03-12     Completed Date:  1999-03-12     Revised Date:  2006-11-15    
Medline Journal Info:
Nlm Unique ID:  7602417     Medline TA:  Gen Pharmacol     Country:  ENGLAND    
Other Details:
Languages:  eng     Pagination:  57-63     Citation Subset:  IM    
Affiliation:
Fuji Gotemba Research Laboratories, Chugai Pharmaceutical Co., Ltd., Shizuoka, Japan. suzukiysy@gt.chugai-pharm.co.jp
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MeSH Terms
Descriptor/Qualifier:
Animals
Anti-Arrhythmia Agents / pharmacology*
Blood Pressure / drug effects
Dogs
Heart / drug effects*,  physiology
Heart Rate / drug effects
Male
Myocardium / metabolism
Oxygen Consumption / drug effects*
Sodium Channels / drug effects
Thiazoles / pharmacology*
Thiazolidines
Chemical
Reg. No./Substance:
0/Anti-Arrhythmia Agents; 0/CP 060S; 0/Sodium Channels; 0/Thiazoles; 0/Thiazolidines

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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