Document Detail


Effect of nicotine on the lower esophageal sphincter. Studies on the mechanism of action.
MedLine Citation:
PMID:  1150020     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Intravenous administration of nicotine sulfate caused a dose-dependent reduction in the lower exophagel sphincter pressure in anesthetized opossums. The maximal reduction in pressure of 85.0 +/- 2.6% was observed with a dose of 50 mug per kg. The effect of 50 mug per kg was not antagonized by bilateral cervical vagotomy, atropine, propranolol or by catecholamine depletion with reserpine. The sphincter relaxation produced by 50 mug per kg of nicotine was antagonized during tachyphylaxis produced by a larger dose (4 mg per kg) of nicotine. Nicotine tachyphylaxis also blocked the vagal-stimulated relaxation of the sphincter. It is suggested that the main action of nicotine on the sphincter in intact animals is caused by its effect on the noncholinergic, nonadrenergic inhibitory neurons which lie in the vagal pathway to the lower esophageal sphincter.
Authors:
S Rattan; R K Goyal
Publication Detail:
Type:  Journal Article; Research Support, U.S. Gov't, P.H.S.    
Journal Detail:
Title:  Gastroenterology     Volume:  69     ISSN:  0016-5085     ISO Abbreviation:  Gastroenterology     Publication Date:  1975 Jul 
Date Detail:
Created Date:  1975-11-06     Completed Date:  1975-11-06     Revised Date:  2006-11-15    
Medline Journal Info:
Nlm Unique ID:  0374630     Medline TA:  Gastroenterology     Country:  UNITED STATES    
Other Details:
Languages:  eng     Pagination:  154-9     Citation Subset:  AIM; IM    
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MeSH Terms
Descriptor/Qualifier:
Animals
Atropine / pharmacology
Electric Stimulation
Esophagogastric Junction / drug effects*
Hexamethonium Compounds / pharmacology
Injections, Intra-Arterial
Injections, Intravenous
Nicotine / administration & dosage,  pharmacology*
Opossums / physiology*
Pressure
Propranolol / pharmacology
Reserpine / pharmacology
Tachyphylaxis
Vagotomy
Chemical
Reg. No./Substance:
0/Hexamethonium Compounds; 50-55-5/Reserpine; 51-55-8/Atropine; 525-66-6/Propranolol; 54-11-5/Nicotine

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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