Document Detail


Drimane sesquiterpenoids from the fungus Aspergillus ustus isolated from the marine sponge Suberites domuncula.
MedLine Citation:
PMID:  19778087     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Seven new drimane sesquiterpenoids (1-3, 6-9), along with the known compounds deoxyuvidin B (4), strobilactone B (5), and RES-1149-2 (10), were obtained from cultures of the fungus Aspergillus ustus, which was isolated from the marine sponge Suberites domuncula. Their structures were established by means of spectroscopic analyses including one- and two-dimensional NMR spectroscopy and high-resolution MS. Compounds 6, 7, and 10 showed cytotoxic activity against a panel of tumor cell lines, including L5178Y, HeLa, and PC12 cells, with 7 being the most active (EC(50) against L5178Y cell line: 0.6 microg/mL).
Authors:
Hongbing Liu; RuAngelie Edrada-Ebel; Rainer Ebel; Yao Wang; Barbara Schulz; Siegfried Draeger; Werner E G Müller; Victor Wray; Wenhan Lin; Peter Proksch
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  Journal of natural products     Volume:  72     ISSN:  1520-6025     ISO Abbreviation:  J. Nat. Prod.     Publication Date:  2009 Sep 
Date Detail:
Created Date:  2009-09-25     Completed Date:  2009-10-21     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  7906882     Medline TA:  J Nat Prod     Country:  United States    
Other Details:
Languages:  eng     Pagination:  1585-8     Citation Subset:  IM    
Affiliation:
Institut fur Pharmazeutische Biologie und Biotechnologie, Heinrich-Heine-Universitat Dusseldorf, Universitatsstrasse 1, Dusseldorf, Germany.
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MeSH Terms
Descriptor/Qualifier:
Animals
Antineoplastic Agents / chemistry,  isolation & purification*,  pharmacology
Aspergillus / chemistry*
Drug Screening Assays, Antitumor
Hela Cells
Humans
Marine Biology
Molecular Structure
Sesquiterpenes / chemistry,  isolation & purification*,  pharmacology
Suberites / microbiology
Chemical
Reg. No./Substance:
0/Antineoplastic Agents; 0/Sesquiterpenes; 0/drimane

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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