Document Detail


Comparative study of the activity of boric, benzene-boronic and methyl-benzene-boronic acids upon respiration, general metabolism and systemic hemodynamics of the anesthetized dog.
MedLine Citation:
PMID:  1174408     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
The authors compared the action of boric, benzene-boronic and p-methyl-benzene-boronic acids on respiration and general metabolism and on systemic hemodynamics of the anesthetized dog. They further investigated the effects on the arterial blood pressure in the rat and on the isolated rabbit heart. In the dogs, the three acids were shown to have no significant action on the systolic, diastolic and mean arterial blood pressures and a slight stimulating action on the differential arterial blood pressure. On the contrary, in the rat, all the acids were hypotensive. This action was dose dependent. In the entire animal, as well as in the isolated rabbit heart, benzene-boronic and p-methyl-benzene-boronic acids depressed the myocardial contractility. Whereas boric acid did not act on the heart contractility in situ in anesthetized dogs, it slightly stimulated the myocardial contractility of the isolated rabbit heart. The two acids seemed to be directly active on the myocardial cell. In the anesthetized dog, cardiac performances were first depressed then stimulated. Both benzene-boronic and p-methyl-benzene-boronic acids were ventilatory depressors: they reduced ventilatory output and rhythm, they first decreased then increased total O2 consumption and CO2 production.
Authors:
Pham-Huu-Chanh; I Sokhan; P Kan
Related Documents :
3601868 - Effect of gizzerosine on acid secretion by isolated mucosal cells of chicken proventric...
2382718 - Luminal cck-releasing factors in the isolated vascularly perfused rat duodenojejunum.
3919168 - Gastric acid secretory function in preterm infants.
17166678 - Inhibition of the gastric h+,k+ -atpase by plectrinone a, a diterpenoid isolated from p...
8723738 - Identification and characterization of limonene metabolites in patients with advanced c...
7859328 - Amphoteric drugs. i. synthesis and antiallergic activity of [4-(diphenylmethoxy)piperid...
Publication Detail:
Type:  Comparative Study; In Vitro; Journal Article    
Journal Detail:
Title:  Arzneimittel-Forschung     Volume:  25     ISSN:  0004-4172     ISO Abbreviation:  Arzneimittelforschung     Publication Date:  1975 Jul 
Date Detail:
Created Date:  1975-12-11     Completed Date:  1975-12-11     Revised Date:  2007-11-15    
Medline Journal Info:
Nlm Unique ID:  0372660     Medline TA:  Arzneimittelforschung     Country:  GERMANY, WEST    
Other Details:
Languages:  eng     Pagination:  1023-8     Citation Subset:  IM; S    
Export Citation:
APA/MLA Format     Download EndNote     Download BibTex
MeSH Terms
Descriptor/Qualifier:
Animals
Benzene Derivatives / pharmacology
Blood Pressure / drug effects
Boric Acids / pharmacology*
Boronic Acids / pharmacology*
Cardiac Output / drug effects
Dogs
Female
Hemodynamics / drug effects*
Male
Myocardial Contraction / drug effects
Oxygen Consumption / drug effects
Rabbits
Rats
Respiration / drug effects*
Toluene / pharmacology
Chemical
Reg. No./Substance:
0/Benzene Derivatives; 0/Boric Acids; 0/Boronic Acids; 108-88-3/Toluene

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


Previous Document:  Structure and actions of saikosaponins isolated from Bupleurum falcatum L. I. Anti-inflammatory acti...
Next Document:  The relevance of the osmolarity of the instillation fluid to the effectiveness and toxicity of drugs...