Document Detail


Combined use of propranolol and nifedipine offers better effects on portal vein nonuniform remodeling in carbon tetrachloride (CCl(4))-induced portal hypertensive rats.
MedLine Citation:
PMID:  19401196     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Portal hypertension is a hemodynamic syndrome due to pathological increase in portal flow and portal pressure. These pathological changes in external flow loads will inevitably cause vascular remodeling in the portal vein, which is usually measured by an opening angle. The present study showed that carbon tetrachloride (CCl(4))-induced portal hypertension fully developed at 8 weeks and the opening angle of portal vein increased progressively in the pathogenesis of intrahepatic portal hypertension which was significantly augmented at 10 weeks. Although portal pressure and portal flow were reduced, treatment with either propranolol or nifedipine alone for 3 weeks did not decrease the augmented opening angle of the portal vein, while combined treatment with propranolol and nifedipine markedly reduced the increased opening angle of the portal vein and endothelial nitric oxide synthase (eNOS) mRNA expression but not inducible nitric oxide synthase (iNOS) mRNA expression. The decreasing effect of propranolol plus nifedipine on the elevated opening angle was significantly weakened by L-arginine and markedly reinforced by N-nitro-l-arginine-mythel-ester (L-NAME). These results indicate that combined use of propranolol and nifedipine ameliorates portal vein remodeling in portal hypertension at least by the nitric oxide-dependent way.
Authors:
Zong-Qi Zhang; Bin Shi; Guo-Qiang Wu; Kai-Rong Qin; Zong-Lai Jiang; Liang Zhu
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't     Date:  2009-05-03
Journal Detail:
Title:  European journal of pharmacology     Volume:  613     ISSN:  1879-0712     ISO Abbreviation:  Eur. J. Pharmacol.     Publication Date:  2009 Jun 
Date Detail:
Created Date:  2009-06-01     Completed Date:  2009-08-28     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  1254354     Medline TA:  Eur J Pharmacol     Country:  Netherlands    
Other Details:
Languages:  eng     Pagination:  108-13     Citation Subset:  IM    
Affiliation:
Department of Gastroenterology, Changzheng Hospital, Second Military Medical University, Shanghai, China.
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MeSH Terms
Descriptor/Qualifier:
Adrenergic beta-Antagonists / pharmacology,  therapeutic use
Animals
Calcium Channel Blockers / pharmacology,  therapeutic use
Carbon Tetrachloride / toxicity*
Drug Combinations
Drug Therapy, Combination
Gene Expression Regulation, Enzymologic / drug effects
Hemodynamics / drug effects
Hypertension, Portal / chemically induced*,  drug therapy,  metabolism,  physiopathology*
Male
Muscle, Smooth / drug effects,  metabolism
Nifedipine / pharmacology*,  therapeutic use
Nitric Oxide Synthase Type II / genetics
Nitric Oxide Synthase Type III / genetics
Portal Vein / drug effects*,  physiopathology*
Propranolol / pharmacology*,  therapeutic use
Rats
Rats, Sprague-Dawley
Chemical
Reg. No./Substance:
0/Adrenergic beta-Antagonists; 0/Calcium Channel Blockers; 0/Drug Combinations; 21829-25-4/Nifedipine; 525-66-6/Propranolol; 56-23-5/Carbon Tetrachloride; EC 1.14.13.39/Nitric Oxide Synthase Type II; EC 1.14.13.39/Nitric Oxide Synthase Type III

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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