Document Detail


Cold exposure decreases the effectiveness of atropine-oxime treatment in organophosphate intoxication in rats and mice.
MedLine Citation:
PMID:  2687080     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
1. The effect of cold environment on the acute toxicity of organophosphates (OP), without and with atropine-oxime treatment, was studied in rats and mice by exposing them to +5 and -5 degrees C temperature. The tested OPs and oximes (given intraperitoneally) were diisopropylfluorophosphate (DFP), isopropyl methylphosphonofluoridate (sarin) and dichlorovinyl phosphate (DDVP), pralidoxime (PAM) and obidoxime. 2. An exposure to low environmental temperature decreased the effectiveness of atropine-oxime therapy in OP poisoned rats and mice, evaluated by means of acute LD50 values. 3. The lowering of environmental temperature did not influence the ability of PAM to reactivate tissue cholinesterase in rats intoxicated by 0.5 x LD50 doses of DFP. 4. The acute toxicity of atropine and oximes was not affected by cold environment in rats, but in mice it was increased by 1.1-2.1 times. 5. The decrease in the effectiveness of atropine-oxime therapy at cold environment may be explained by the observation that the cold temperature sensitizes the animals to the inhibition of brain acetylcholinesterase by OP.
Authors:
E Kaliste-Korhonen; R Ryhänen; P Ylitalo; O Hänninen
Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  General pharmacology     Volume:  20     ISSN:  0306-3623     ISO Abbreviation:  Gen. Pharmacol.     Publication Date:  1989  
Date Detail:
Created Date:  1990-01-25     Completed Date:  1990-01-25     Revised Date:  2008-11-21    
Medline Journal Info:
Nlm Unique ID:  7602417     Medline TA:  Gen Pharmacol     Country:  ENGLAND    
Other Details:
Languages:  eng     Pagination:  805-9     Citation Subset:  IM    
Affiliation:
Department of Physiology, University of Kuopio, Finland.
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MeSH Terms
Descriptor/Qualifier:
Animals
Antidotes*
Atropine / pharmacology*
Carboxylic Ester Hydrolases / antagonists & inhibitors,  metabolism
Cholinesterase Reactivators
Cold Temperature
Enzyme Reactivators
Isoflurophate / poisoning
Lethal Dose 50
Mice
Obidoxime Chloride / pharmacology
Organophosphorus Compounds / poisoning*
Oximes / pharmacology*
Pralidoxime Compounds / pharmacology
Rats
Rats, Inbred F344
Chemical
Reg. No./Substance:
0/Antidotes; 0/Cholinesterase Reactivators; 0/Enzyme Reactivators; 0/Organophosphorus Compounds; 0/Oximes; 0/Pralidoxime Compounds; 114-90-9/Obidoxime Chloride; 51-55-8/Atropine; 55-91-4/Isoflurophate; 6735-59-7/pralidoxime; EC 3.1.1.-/Carboxylic Ester Hydrolases

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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