Document Detail


Colchicine myopathy and neuromyopathy: two cases with different characteristics.
MedLine Citation:
PMID:  20661070     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Colchicine, a long established anti-inflammatory agent now used in several rheumatologic conditions, acts by inhibiting microtubular polymerization, as it binds equimolarly to tubulin molecules. Cytoskeletal microtubules are crucial in processes of cell viability, such as mitosis and intracellular vesicle motility.Gastrointestinal side effects are quite common and often minor in nature or duration, whereas neuromuscular toxicity is rare. We report 2 cases of colchicine myopathy in the context of very different clinical settings.
Authors:
Luca Cantarini; Nila Volpi; Mauro Galeazzi; Teresa Giani; Francesca Fanti; Orso Maria Lucherini; Margherita Aglianò; Carlo Alessandrini; Fabio Giannini; Stefania Magi; Giuseppe Greco; Cosima Tatiana Baldari; Rolando Cimaz
Publication Detail:
Type:  Case Reports; Journal Article    
Journal Detail:
Title:  Journal of clinical rheumatology : practical reports on rheumatic & musculoskeletal diseases     Volume:  16     ISSN:  1536-7355     ISO Abbreviation:  J Clin Rheumatol     Publication Date:  2010 Aug 
Date Detail:
Created Date:  2010-07-27     Completed Date:  2010-12-16     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  9518034     Medline TA:  J Clin Rheumatol     Country:  United States    
Other Details:
Languages:  eng     Pagination:  229-32     Citation Subset:  IM    
Affiliation:
Interdepartmental Research Center of Systemic Autoimmune and Autoinflammatory Diseases, Unit of Rheumatology, Policlinico Le Scotte, University of Siena, Siena, Italy. cantariniluca@hotmail.com
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MeSH Terms
Descriptor/Qualifier:
Adolescent
Arthritis, Gouty / drug therapy
Colchicine / adverse effects*,  metabolism,  therapeutic use
Cytochrome P-450 CYP3A / metabolism
Familial Mediterranean Fever / drug therapy
Female
Humans
Male
Middle Aged
Muscle Weakness / chemically induced,  diagnosis
Muscular Diseases / chemically induced*,  diagnosis
P-Glycoprotein / metabolism
Tubulin Modulators / adverse effects*,  metabolism,  therapeutic use
Chemical
Reg. No./Substance:
0/P-Glycoprotein; 0/Tubulin Modulators; 64-86-8/Colchicine; EC 1.14.13.67/CYP3A4 protein, human; EC 1.14.14.1/Cytochrome P-450 CYP3A

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