Document Detail


Cardiac electrophysiological actions and interactions of ethanol, cocaine, and the metabolite ethylcocaine.
MedLine Citation:
PMID:  9817212     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
The influence of ethanol on the actions of cocaine and ethylcocaine on rat sinoatrial preparations was studied. Ethanol did not modify the depressant effect of cocaine or ethylcocaine on sinoatrial rate (SR) in preparations with spontaneous activity. Cocaine produced sinoatrial block only in the presence of ethanol, and the latter accentuated the sinoatrial block produced by ethylcocaine. Ethanol did not modify the depressant effect of cocaine or ethylcocaine on membrane potentials of atrial fibers in preparations driven at a constant rate. In conclusion, ethanol, in a concentration that did not by itself affect SR or produce sinoatrial block, accentuated the effects of cocaine and ethylcocaine on sinoatrial conduction, without modifying the effects on SR. It is proposed that the accentuation of the block was the consequence of the combination of a depressant action on the fast sodium system and a deterioration of the cell-to-cell coupling.
Authors:
A K Jain; R G Carpentier
Publication Detail:
Type:  Comparative Study; In Vitro; Journal Article; Research Support, U.S. Gov't, P.H.S.    
Journal Detail:
Title:  Journal of electrocardiology     Volume:  31     ISSN:  0022-0736     ISO Abbreviation:  J Electrocardiol     Publication Date:  1998 Oct 
Date Detail:
Created Date:  1999-01-21     Completed Date:  1999-01-21     Revised Date:  2009-11-11    
Medline Journal Info:
Nlm Unique ID:  0153605     Medline TA:  J Electrocardiol     Country:  UNITED STATES    
Other Details:
Languages:  eng     Pagination:  293-302     Citation Subset:  IM    
Affiliation:
Department of Physiology and Biophysics, College of Medicine, Howard University, Washington, DC 20059, USA.
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MeSH Terms
Descriptor/Qualifier:
Action Potentials / drug effects
Animals
Cocaine / analogs & derivatives*,  pharmacology*
Drug Interactions
Electrophysiology
Ethanol / pharmacology*
Male
Microelectrodes
Rats
Rats, Sprague-Dawley
Sinoatrial Block / chemically induced*,  physiopathology
Sinoatrial Node / drug effects*,  physiopathology
Grant Support
ID/Acronym/Agency:
S06GM8016/GM/NIGMS NIH HHS
Chemical
Reg. No./Substance:
50-36-2/Cocaine; 529-38-4/cocaethylene; 64-17-5/Ethanol

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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