Document Detail


Antitumor efficacy of poly(dimer acid-dodecanedioic acid) copolymer in mice bearing Sarcoma-180 tumor.
MedLine Citation:
PMID:  17387591     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
The drug release profiles of poly(dimer acid-dodecanedioic acid) P(DA-DDDA) copolymer containing 5% adriamycin hydrochloride (ADM) in vitro were evaluated. The biocompatibility of P(DA-DDDA) under mice skin was also evaluated, macroscopic observation and microscopic analysis demonstrated that the copolymer is biocompatible and well tolerated in vivo. Antitumor efficacy of P(DA-DDDA) copolymers containing 5% adriamycin hydrochloride (ADM) implanted subcutaneously in mice bearing Sarcoma-180 tumor exhibited increased volume doubling time (VDT) (31 +/- 1.5 days) compared to plain subcutaneous injection of ADM (7 +/- 0.9 days). The studies suggest that P(DA-DDDA) copolymer as an effective carrier for antineoplastic drug like adriamycin hydrochloride has a very good prospect in the treatment of noumenon tumors.
Authors:
Wen-Xun Guo; Zongli Shi; Fan-Bing Zeng; Kui Liang; Xian-Hong Chen; Yong-Ping Ai; Min Fang; Xiao Sun; Zhi Zhang; Li-Xin Hu
Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't     Date:  2007-03-27
Journal Detail:
Title:  Journal of materials science. Materials in medicine     Volume:  18     ISSN:  0957-4530     ISO Abbreviation:  J Mater Sci Mater Med     Publication Date:  2007 Aug 
Date Detail:
Created Date:  2007-07-04     Completed Date:  2007-10-19     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  9013087     Medline TA:  J Mater Sci Mater Med     Country:  United States    
Other Details:
Languages:  eng     Pagination:  1515-20     Citation Subset:  IM    
Affiliation:
College of Materials Science and Engineering, Hunan University, Changsha, Hunan 410082, P.R. China. guowenxun@126.com
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MeSH Terms
Descriptor/Qualifier:
Animals
Antibiotics, Antineoplastic / administration & dosage*,  chemistry,  pharmacokinetics
Cell Line, Tumor
Cell Survival / drug effects
Delayed-Action Preparations / administration & dosage*,  chemistry,  pharmacokinetics
Dicarboxylic Acids / administration & dosage*,  chemistry,  pharmacokinetics
Diffusion
Doxorubicin / administration & dosage*,  chemistry,  pharmacokinetics
Drug Compounding / methods
Drug Implants
Injections, Subcutaneous
Materials Testing
Mice
Polymers / administration & dosage*,  chemistry,  pharmacokinetics
Sarcoma / drug therapy*,  pathology*
Treatment Outcome
Chemical
Reg. No./Substance:
0/Antibiotics, Antineoplastic; 0/Delayed-Action Preparations; 0/Dicarboxylic Acids; 0/Drug Implants; 0/Polymers; 0/poly(dimer acid-dodecanedioic acid) copolymer; 23214-92-8/Doxorubicin

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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