Document Detail


Anandamide protects from low serum-induced apoptosis via its degradation to ethanolamine.
MedLine Citation:
PMID:  17227767     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Anandamide (AEA) is a lipid molecule belonging to the family of endocannabinoids. Various studies report neuroprotective activity of AEA against toxic insults, such as ischemic conditions and excitotoxicity, whereas some show that AEA has pro-apoptotic effects. Here we have shown that AEA confers a protective activity in N18TG2 murine neuroblastoma cells subjected to low serum-induced apoptosis. We have demonstrated that the protection from apoptosis by AEA is not mediated via the CB1 receptor, the CB2 receptor, or the vanilloid receptor 1. Interestingly, breakdown of AEA by fatty acid amide hydrolase is required for the protective effect of AEA. Furthermore, the ethanolamine (EA) generated in this reaction is the metabolite responsible for the protective response. The elevation in the levels of reactive oxygen species during low serum-induced apoptosis is not affected by AEA or EA. On the other hand, AEA and EA reduce caspase 3/7 activity, and AEA attenuates the cleavage of PARP-1. Taken together, our results demonstrate a role for AEA and EA in the protection against low serum-induced apoptosis.
Authors:
Devorah Matas; Ana Juknat; Maciej Pietr; Yael Klin; Zvi Vogel
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Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't     Date:  2007-01-16
Journal Detail:
Title:  The Journal of biological chemistry     Volume:  282     ISSN:  0021-9258     ISO Abbreviation:  J. Biol. Chem.     Publication Date:  2007 Mar 
Date Detail:
Created Date:  2007-03-12     Completed Date:  2007-04-24     Revised Date:  -    
Medline Journal Info:
Nlm Unique ID:  2985121R     Medline TA:  J Biol Chem     Country:  United States    
Other Details:
Languages:  eng     Pagination:  7885-92     Citation Subset:  IM    
Affiliation:
Department of Neurobiology, Weizmann Institute of Science, 76100 Rehovot, Israel.
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MeSH Terms
Descriptor/Qualifier:
Amidohydrolases / metabolism
Animals
Apoptosis*
Arachidonic Acids / pharmacology*
Caspase 3 / metabolism
Caspase 7 / metabolism
Cell Line, Tumor
DNA Fragmentation
Dose-Response Relationship, Drug
Ethanolamine / metabolism*
Flow Cytometry
Ischemia
Mice
Neuroblastoma / metabolism
Polyunsaturated Alkamides / pharmacology*
Reactive Oxygen Species
Receptors, Cannabinoid / metabolism
TRPV Cation Channels / metabolism
Chemical
Reg. No./Substance:
0/Arachidonic Acids; 0/Polyunsaturated Alkamides; 0/Reactive Oxygen Species; 0/Receptors, Cannabinoid; 0/TRPV Cation Channels; 141-43-5/Ethanolamine; 94421-68-8/anandamide; EC 3.4.22.-/Caspase 3; EC 3.4.22.-/Caspase 7; EC 3.5.-/Amidohydrolases; EC 3.5.1.-/fatty-acid amide hydrolase

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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