Document Detail


Alleviation of cocaine-induced coronary vasoconstriction by nitroglycerin.
MedLine Citation:
PMID:  1906905     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Cocaine induces vasoconstriction of epicardial coronary arteries in patients with and without coronary artery disease, and this vasoconstriction is particularly marked in segments narrowed by atherosclerosis. To assess the effect of nitroglycerin on cocaine-induced coronary vasoconstriction, computer-assisted quantitative analysis was performed on non-diseased and diseased coronary artery segments in 23 patients (18 men, 5 women, aged 43 to 65 years) 1) at baseline, 2) after administration of intranasal saline solution (in 8 patients) or 2 mg/kg of cocaine (in 15 patients), and then 3) after administration of sublingual placebo (in 6 patients) or 0.4 or 0.8 mg of nitroglycerin (in 9 patients) in the 15 patients given cocaine. In response to cocaine administration, coronary artery cross-sectional area decreased 22 +/- 7% (mean +/- SD) in non-diseased segments (p less than 0.05) and 45 +/- 18% in diseased segments (p less than 0.02). The magnitude of vasoconstriction was greater (p = 0.01) in the diseased segments. Sublingual nitroglycerin abolished the vasoconstriction in both non-diseased and diseased segments. Thus, nitroglycerin alleviates cocaine-induced vasoconstriction in patients with coronary artery disease.
Authors:
W C Brogan; R A Lange; A S Kim; D J Moliterno; L D Hillis
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Publication Detail:
Type:  Clinical Trial; Controlled Clinical Trial; Journal Article; Research Support, Non-U.S. Gov't; Research Support, U.S. Gov't, P.H.S.    
Journal Detail:
Title:  Journal of the American College of Cardiology     Volume:  18     ISSN:  0735-1097     ISO Abbreviation:  J. Am. Coll. Cardiol.     Publication Date:  1991 Aug 
Date Detail:
Created Date:  1991-08-26     Completed Date:  1991-08-26     Revised Date:  2007-11-15    
Medline Journal Info:
Nlm Unique ID:  8301365     Medline TA:  J Am Coll Cardiol     Country:  UNITED STATES    
Other Details:
Languages:  eng     Pagination:  581-6     Citation Subset:  AIM; IM    
Affiliation:
Department of Internal Medicine, University of Texas Southwestern Medical Center, Dallas 75235.
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MeSH Terms
Descriptor/Qualifier:
Administration, Intranasal
Administration, Sublingual
Aged
Cocaine / administration & dosage,  adverse effects*
Coronary Angiography
Coronary Artery Disease / physiopathology
Coronary Vessels / drug effects*
Female
Heart Catheterization
Humans
Male
Middle Aged
Nitroglycerin / administration & dosage,  therapeutic use*
Vasoconstriction / drug effects*
Grant Support
ID/Acronym/Agency:
HL-17669/HL/NHLBI NIH HHS
Chemical
Reg. No./Substance:
50-36-2/Cocaine; 55-63-0/Nitroglycerin

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


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