Document Detail


Aldosterone receptor antagonists: focus on eplerenone.
MedLine Citation:
PMID:  12624573     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Despite the development of hypertension treatment guidelines, blood pressure control in the general population remains inadequate, indicating the need for ongoing re-evaluation of treatment strategies to further improve blood pressure control. Hypertension results from alterations in cardiac output and/or peripheral resistance. The renin-angiotensin-aldosterone system may be responsible, at least in part, for these alterations. Despite pharmacologic intervention with angiotensin-converting enzyme inhibitors and angiotensin type-1 receptor antagonists, aldosterone continues to be produced. Therapeutic modalities for treating hypertension directed toward antagonizing aldosterone might more effectively control blood pressure. Eplerenone, a new selective aldosterone receptor antagonist, recently received approval from the US Food and Drug Administration for the treatment of hypertension, either alone or in combination with other antihypertensive agents. The objective of this review is to summarize the renin-angiotensin-aldosterone system, emphasizing the role for aldosterone antagonism in the management of hypertension, with a focus on eplerenone.
Authors:
Robert E Lamb; Jon Folstad
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Publication Detail:
Type:  Journal Article; Review    
Journal Detail:
Title:  Progress in cardiovascular nursing     Volume:  18     ISSN:  0889-7204     ISO Abbreviation:  Prog Cardiovasc Nurs     Publication Date:  2003  
Date Detail:
Created Date:  2003-03-07     Completed Date:  2003-05-15     Revised Date:  2005-11-16    
Medline Journal Info:
Nlm Unique ID:  8704064     Medline TA:  Prog Cardiovasc Nurs     Country:  United States    
Other Details:
Languages:  eng     Pagination:  54-9     Citation Subset:  IM; N    
Copyright Information:
Copyright 2003 CHF, Inc.
Affiliation:
AstraZeneca LP, 725 Chesterbrook Boulevard, Wayne, PA 19087, USA. robert.lamb@astrazeneca.com
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MeSH Terms
Descriptor/Qualifier:
Aldosterone Antagonists / standards,  therapeutic use
Antihypertensive Agents / antagonists & inhibitors,  standards,  therapeutic use
Blood Pressure / drug effects
Cardiac Output / drug effects
Humans
Receptors, Aldosterone / antagonists & inhibitors*,  therapeutic use
Renin-Angiotensin System / drug effects
Spironolactone / analogs & derivatives*,  antagonists & inhibitors,  standards,  therapeutic use
United States
Vascular Resistance / drug effects
Chemical
Reg. No./Substance:
0/Aldosterone Antagonists; 0/Antihypertensive Agents; 0/Receptors, Aldosterone; 0/eplerenone; 52-01-7/Spironolactone

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