Document Detail


Activation of calpain I converts excitotoxic neuron death into a caspase-independent cell death.
MedLine Citation:
PMID:  10828077     Owner:  NLM     Status:  MEDLINE    
Abstract/OtherAbstract:
Glutamate receptor overactivation contributes to neuron death after stroke, trauma, and epileptic seizures. Exposure of cultured rat hippocampal neurons to the selective glutamate receptor agonist N-methyl-d-aspartate (300 microm, 5 min) or to the apoptosis-inducing protein kinase inhibitor staurosporine (300 nm) induced a delayed neuron death. In both cases, neuron death was preceded by the mitochondrial release of the pro-apoptotic factor cytochrome c. Unlike staurosporine, the N-methyl-d-aspartate-induced release of cytochrome c did not lead to significant activation of caspase-3, the main caspase involved in the execution of neuronal apoptosis. In contrast, activation of the Ca(2+)-activated neutral protease calpain I was readily detectable after the exposure to N-methyl-d-aspartate. In a neuronal cell-free apoptosis system, calpain I prevented the ability of cytochrome c to activate the caspase cascade by inhibiting the processing of procaspase-3 and -9 into their active subunits. In the hippocampal neuron cultures, the inhibition of calpain activity restored caspase-3-like protease activity after an exposure to N-methyl-d-aspartate. Our data demonstrate the existence of signal transduction pathways that prevent the entry of cells into a caspase-dependent cell death program after the mitochondrial release of cytochrome c.
Authors:
S Lankiewicz; C Marc Luetjens; N Truc Bui; A J Krohn; M Poppe; G M Cole; T C Saido; J H Prehn
Related Documents :
10869477 - Upregulation of the expression of fas antigen and fas ligand in a human submandibular g...
11599307 - Preclinical development of neurosteroids as neuroprotective agents for the treatment of...
10652467 - Role of the common cytokine receptor gamma chain (gammac) in thymocyte selection.
15784847 - The neurotransmitter noradrenaline rescues septal cholinergic neurons in culture from d...
9463487 - Ivermectin: a positive allosteric effector of the alpha7 neuronal nicotinic acetylcholi...
9016917 - In vivo blockade of thalamic gaba(b) receptors increases excitatory amino-acid levels.
Publication Detail:
Type:  Journal Article; Research Support, Non-U.S. Gov't    
Journal Detail:
Title:  The Journal of biological chemistry     Volume:  275     ISSN:  0021-9258     ISO Abbreviation:  J. Biol. Chem.     Publication Date:  2000 Jun 
Date Detail:
Created Date:  2000-07-11     Completed Date:  2000-07-11     Revised Date:  2006-11-15    
Medline Journal Info:
Nlm Unique ID:  2985121R     Medline TA:  J Biol Chem     Country:  UNITED STATES    
Other Details:
Languages:  eng     Pagination:  17064-71     Citation Subset:  IM    
Affiliation:
Interdisciplinary Center for Clinical Research (IZKF), Research Group "Apoptosis and Cell Death," Westphalian Wilhelms University, D-48149 Münster, Germany.
Export Citation:
APA/MLA Format     Download EndNote     Download BibTex
MeSH Terms
Descriptor/Qualifier:
Animals
Apoptosis / drug effects*
Calpain / metabolism*
Caspases / metabolism
Cells, Cultured
Cytochrome c Group / metabolism
Enzyme Activation
Hippocampus / drug effects,  enzymology
Microscopy, Fluorescence
Mitochondria / drug effects,  enzymology
N-Methylaspartate / pharmacology*
Neurons / cytology,  drug effects*,  enzymology
Rats
Chemical
Reg. No./Substance:
0/Cytochrome c Group; 6384-92-5/N-Methylaspartate; EC 3.4.22.-/Calpain; EC 3.4.22.-/Caspases

From MEDLINE®/PubMed®, a database of the U.S. National Library of Medicine


Previous Document:  Regulation of receptor-mediated protein kinase C membrane trafficking by autophosphorylation.
Next Document:  Apolipoprotein A-I: structure-function relationships.